| Article ID ▲/▼ | Title ▲/▼ | Authors ▲/▼ | Journal | Year ▲/▼ | DOI | Records |
|---|
| cpdart0001 | Accumulation of arginine-rich cell-penetrating peptides in tumors and the potential for anticancer drug delivery in vivo. | Nakase, Ikuhiko; Konishi, Yusuke; Ueda, Masashi; Saji, Hideo; Futaki, Shiroh | Journal of controlled release : official journal of the Controlled Release Society | 2012 | | 1 |
| cpdart0005 | Design and biological evaluation of cell-penetrating peptide-doxorubicin conjugates as prodrugs. | Nasrolahi Shirazi, Amir; Tiwari, Rakesh; Chhikara, Bhupender S; Mandal, Dindyal; Parang, Keykavous | Molecular pharmaceutics | 2013 | | 2 |
| cpdart0012 | Controlled release of free doxorubicin from peptide-drug conjugates by drug loading. | Chen, Zhipeng; Zhang, Pengcheng; Cheetham, Andrew G; Moon, Jae Hyon; Moxley, James W Jr; Lin, Yi-an; Cui, Honggang | Journal of controlled release : official journal of the Controlled Release Society | 2014 | | 3 |
| cpdart0014 | Cell penetrating peptides as efficient nanocarriers for delivery of antifungal compound, natamycin for the treatment of fungal keratitis. | Jain, Aastha; Shah, Sushmita G; Chugh, Archana | Pharmaceutical research | 2015 | | 1 |
| cpdart0015 | Activable Cell-Penetrating Peptide Conjugated Prodrug for Tumor Targeted Drug Delivery. | Cheng, Hong; Zhu, Jing-Yi; Xu, Xiao-Ding; Qiu, Wen-Xiu; Lei, Qi; Han, Kai; Cheng, Yin-Jia; Zhang, Xian-Zheng | ACS Applied Materials & Interfaces | 2015 | | 1 |
| cpdart0016 | Dual-targeting hybrid peptide-conjugated doxorubicin for drug resistance reversal in breast cancer. | Sheng, Yuan; You, Yiwen; Chen, Yun | International Journal of Pharmaceutics | 2016 | | 1 |
| cpdart0020 | BH3 mimetics derived from Bim-BH3 domain core region show PTP1B inhibitory activity. | Lu, Xiao; Wu, Lijuan; Liu, Xiaochun; Wang, Shulin; Zhang, Chuanliang | Bioorganic and Medicinal Chemistry Letters | 2019 | | 1 |
| cpdart0021 | Increasing the potential of cell-penetrating peptides for cancer therapy using a new pentagonal scaffold. | Duarte, Diana; Fraga, Alexandra G.; Pedrosa, Jorge; Martel, Fátima; Vale, Nuno | European Journal of Pharmacology | 2019 | | 6 |
| cpdart0023 | Novel peptide conjugates for tumor-specific chemotherapy. | Langer, Michael; Kratz, Felix; Rothen-Rutishauser, Barbara; Wunderli-Allenspach, Heidi; Beck-Sickinger, Annette G. | Journal of Medicinal Chemistry | 2001 | | 2 |
| cpdart0025 | Peptide-Drug Conjugate Linked via a Disulfide Bond for Kidney Targeted Drug Delivery | Geng, Qian; Sun, Xun; Gong, Tao; Zhang, Zhi-Rong | Bioconjugate Chemistry | 2012 | | 2 |
| cpdart0026 | Cancer chemotherapy based on targeting of cytotoxic peptide conjugates to their receptors on tumors | Schally, Andrew V.; Nagy, Attila | European Journal of Endocrinology | 1999 | | 1 |
| cpdart0027 | Design, synthesis and biological evaluation of peptide-NSAID conjugates for targeted cancer therapy | Shokri, Bahareh; Zarghi, Afshin; Shahhoseini, Soraya; Mohammadi, Reza; Kobarfard, Farzad | Archiv der Pharmazie | 2019 | | 8 |
| cpdart0028 | Synthesis and anti-cancer evaluation of folic acid-peptide- paclitaxel conjugates for addressing drug resistance | Dai, Yuxuan; Cai, Xingguang; Bi, Xinzhou; Liu, Chunxia; Yue, Na; Zhu, Ying; Zhou, Jiaqi; Fu, Mian; Huang, Wenlong; Qian, Hai | European Journal of Medicinal Chemistry | 2019 | | 7 |
| cpdart0029 | Synthesis and biological evaluation of a novel series of curcumin-peptide derivatives as PepT1-mediated transport drugs | Zhang, Jiyun; Wen, Hongmei; Shen, Fei; Wang, Xinzhi; Shan, Chenxiao; Chai, Chuan; Liu, Jian; Li, Wei | Bioorganic Chemistry | 2019 | | 20 |
| cpdart0030 | N-Methyl-N-phenylvinylsulfonamides for Cysteine-Selective Conjugation | Huang, Rong; Li, Zhihong; Sheng, Yao; Yu, Jianghui; Wu, Yue; Zhan, Yuexiong; Chen, Hongli; Jiang, Biao | Organic Letters | 2018 | | 12 |
| cpdart0031 | Chemoselective Peptide Modification via Photocatalytic Tryptophan β-Position Conjugation | Yu, Younong; Zhang, Li-Kang; Buevich, Alexei V.; Li, Guoqing; Tang, Haiqun; Vachal, Petr; Colletti, Steven L.; Shi, Zhi-Cai | Journal of the American Chemical Society | 2018 | | 20 |
| cpdart0032 | Effect of low charge and high hydrophobicity on antimicrobial activity of the quinazolinone-peptide conjugates | Rakesh, Kadallipura Puttaswamy; Ramesh, Suhas; Shivakumar; Gowda, Dase Channe | Russian Journal of Bioorganic Chemistry | 2018 | | 20 |
| cpdart0033 | In vitro biological evaluation of new antimycobacterial salicylanilide-tuftsin conjugates | European Journal of Medicinal Chemistry | European Journal of Medicinal Chemistry | 2017 | | 22 |
| cpdart0034 | Enhancing the Potency of Nalidixic Acid toward a Bacterial DNA Gyrase with Conjugated Peptides | Ahmed, Marya; Kelley, Shana O. | ACS Chemical Biology | 2017 | | 5 |
| cpdart0035 | Biological characterization of novel nitroimidazole-peptide conjugates in vitro and in vivo | Bergmann, Ralf; Splith, Katrin; Pietzsch, Jens; Bachmann, Michael; Neundorf, Ines | Journal of Peptide Science | 2017 | | 4 |
| cpdart0036 | Peptide Conjugates of Benzene Carboxylic Acids as Agonists and Antagonists of Amylin Aggregation | Profit, Adam A.; Vedad, Jayson; Desamero, Ruel Z. B. | Bioconjugate Chemistry | 2017 | | 9 |
| cpdart0037 | Truncated Autoinducing Peptide Conjugates Selectively Recognize and Kill Staphylococcus aureus | Tsuchikama, Kyoji; Shimamoto, Yasuhiro; Anami, Yasuaki | ACS Infectious Diseases | 2017 | | 13 |
| cpdart0038 | Cyclic peptide conjugate of curcumin and doxorubicin as an anticancer agent | Darwish, Shaban; Mozaffari, Saghar; Parang, Keykavous; Tiwari, Rakesh | Tetrahedron Letters | 2017 | | 2 |
| cpdart0039 | Designing Hybrid Antibiotic Peptide Conjugates To Cross Bacterial Membranes | Deshayes, Stephanie; Xian, Wujing; Schmidt, Nathan W.; Kordbacheh, Shadi; Lieng, Juelline; Wang, Jennifer; Zarmer, Sandra; Germain, Samantha St.; Voyen, Laura; Thulin, Julia; Wong, Gerard C. L.; Kasko, Andrea M. | Bioconjugate Chemistry | 2017 | | 5 |
| cpdart0040 | Microwave Energy in Ugi Four-Component Reaction (Ugi-4CR): Expedient Synthesis of Steroid-Peptide Conjugates Based on Aminosteroids - An Important Class of Hybrid Systems | Borah, Preetismita; Chowdhury, Pritish; Begum, Ashma | Current Organic Synthesis | 2017 | | 5 |
| cpdart0041 | Cell-penetrating conjugates of pentaglutamylated methotrexate as potential anticancer drugs against resistant tumor cells | Szabo, Ildiko; Orban, Erika; Schlosser, Gitta; Hudecz, Ferenc; Banoczi, Zoltan | European Journal of Medicinal Chemistry | 2016 | | 7 |
| cpdart0042 | Design, synthesis, and evaluation of Trolox-conjugated amyloid-β C-terminal peptides for therapeutic intervention in an in vitro model of Alzheimer’s disease | Arai, Takuya; Ohno, Akiko; Kazunori, Mori; Kakizawa, Taeko; Kuwata, Hiroshi; Ozawa, Toshihiko; Shibanuma, Motoko; Hara, Shuntaro; Ishida, Seiichi; Kurihara, Masaaki; Miyata, Naoki; Nakagawa, Hidehiko; Fukuhara, Kiyoshi | Bioorganic & Medicinal Chemistry | 2016 | | 11 |
| cpdart0043 | Delivering aminopyridine ligands into cancer cells through conjugation to the cell-penetrating peptide BP16 | Soler, M.; Gonzalez-Bartulos, M.; Figueras, E.; Massaguer, A.; Feliu, L.; Planas, M.; Ribas, X.; Costas, M. | Organic & Biomolecular Chemistry | 2016 | | 10 |
| cpdart0044 | Dual Targeting of Intracellular Pathogenic Bacteria with a Cleavable Conjugate of Kanamycin and an Antibacterial Cell-Penetrating Peptide | Brezden, Anna; Mohamed, Mohamed F.; Nepal, Manish; Harwood, John S.; Kuriakose, Jerrin; Seleem, Mohamed N.; Chmielewski, Jean | Journal of the American Chemical Society | 2016 | | 2 |
| cpdart0045 | An effective conjugation strategy for designing short peptide-based HIV-1 fusion inhibitors | Liang, Guodong; Wang, Huixin; Chong, Huihui; Cheng, Siqi; Jiang, Xifeng; He, Yuxian; Wang, Chao; Liu, Keliang | Organic & Biomolecular Chemistry | 2016 | | 5 |
| cpdart0046 | Peptide-assisted enhancement of inhibitory effects of small molecular inhibitors for kinases | Wang, Wei; Hirano, Yoshinori; Uzawa, Takanori; Taiji, Makoto; Ito, Yoshihiro | Bulletin of the Chemical Society of Japan | 2016 | | 1 |
| cpdart0047 | Linker dependent chirality of solvent induced self-assembled structures of porphyrin–α-helical peptide conjugates | Biscaglia, Francesca; Frezza, Elisa; Zurlo, Enrico; Gobbo, Marina | Organic & Biomolecular Chemistry | 2016 | | 10 |
| cpdart0048 | Design and synthesis of peptide conjugates of phosphoramide mustard as prodrugs activated by prostate-specific antigen | Wu, Xinghua; Hu, Longqin | Bioorganic & Medicinal Chemistry | 2016 | | 6 |
| cpdart0050 | Intracellular Generation of a Diterpene-Peptide Conjugate that Inhibits 14-3-3-Mediated Interactions | Parvatkar, Prakash; Kato, Nobuo; Uesugi, Motonari; Sato, Shin-ichi; Ohkanda, Junko | Journal of the American Chemical Society | 2015 | | 3 |
| cpdart0051 | Synthesis, drug release, and biological evaluation of new anticancer drug-bioconjugates containing somatostatin backbone cyclic analog as a targeting moiety | Redko, Boris; Ragozin, Elena; Andreii, Bazylevich; Helena, Tuchinsky; Amnon, Albeck; Talia, Shekhter Zahavi; Mor, Oron-Herman; Genady, Kostenich; Gary, Gellerman | Biopolymers | 2015 | | 5 |
| cpdart0052 | Synthesis of a New Peptide-Coumarin Conjugate: A Potential Agent against Cryptococcosis | Ferreira, Soraya Z.; Carneiro, Hellem C.; Lara, Hugo A.; Alves, Rosemeire B.; Resende, Jarbas M.; Oliveira, Heloisa M.; Silva, Luciana M.; Santos, Daniel A.; Freitas, Rossimiriam P. | ACS Medicinal Chemistry Letters | 2015 | | 1 |
| cpdart0053 | Synthesis of Tridecaptin-Antibiotic Conjugates with in Vivo Activity against Gram-Negative Bacteria | Cochrane, Stephen A.; Li, Xuefeng; He, Sisi; Yu, Min; Wu, Min; Vederas, John C. | Journal of Medicinal Chemistry | 2015 | | 6 |
| cpdart0055 | Aminocatalysis-Mediated on-Resin Ugi Reactions: Application in the Solid-Phase Synthesis of N-Substituted and Tetrazolo Lipopeptides and Peptidosteroids | Morales, Fidel E.; Garay, Hilda E.; Munoz, Daniela F.; Augusto, Yarelys E.; Otero-Gonzalez, Anselmo J.; Reyes Acosta, Osvaldo; Rivera, Daniel G. | Organic Letters | 2015 | | 14 |
| cpdart0056 | Synthesis and Activity of 6″-Deoxy-6″-thio-α-GalCer and Peptide Conjugates | Compton, Benjamin J.; Tang, Ching-wen; Johnston, Karen A.; Osmond, Taryn L.; Hayman, Colin M.; Larsen, David S.; Hermans, Ian F.; Painter, Gavin F. | Organic Letters | 2015 | | 2 |
| cpdart0057 | Efficient synthesis of peptide and protein functionalized pyrrole-imidazole polyamides using native chemical ligation | Janssen, Brian M. G.; van Ommeren, Sven P. F. I.; Merkx, Maarten | International Journal of Molecular Sciences | 2015 | | 2 |
| cpdart0058 | Tetrapeptide-coumarin conjugate 3D networks based on hydrogen-bonded charge transfer complexes: gel formation and dye release | Guo, Zongxia; Gong, Ruiying; Jiang, Yi; Wan, Xiaobo | Soft Matter | 2015 | | 2 |
| cpdart0059 | Enhancing Accumulation and Penetration of HPMA Copolymer-Doxorubicin Conjugates in 2D and 3D Prostate Cancer Cells via iRGD Conjugation with an MMP-2 Cleavable Spacer | Peng, Zheng-Hong; Kopecek, Jindrich | Journal of the American Chemical Society | 2015 | | 1 |
| cpdart0060 | Synthesis of bisarylethyne-peptide conjugates | Strack, Martin; Langklotz, Sina; Bandow, Julia E.; Metzler-Nolte, Nils; Bauke Albada, H. | Organic Chemistry Frontiers | 2015 | | 2 |
| cpdart0061 | Solid-phase-based synthesis of ureidopyrimidinone-peptide conjugates for supramolecular biomaterials | de Feijter, Isja; Goor, Olga J. G. M.; Hendrikse, Simone I. S.; Comellas-Aragones, Marta; Soentjens, Serge H. M.; Zaccaria, Sabrina; Fransen, Peter P. K. H.; Peeters, Joris W.; Milroy, Lech-Gustav; Dankers, Patricia Y. W. | Synlett | 2015 | | 31 |
| cpdart0062 | Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activity | Govdi, Anastasiya I.; Sokolova, Nadezda V.; Sorokina, Irina V.; Baev, Dmitry S.; Tolstikova, Tatyana G.; Mamatyuk, Victor I.; Fadeev, Dmitry S.; Vasilevsky, Sergey F.; Nenajdenko, Valentine G. | MedChemComm | 2015 | | 7 |
| cpdart0063 | Solid-phase synthesis of peptide conjugates derived from the antimicrobial cyclic decapeptide BPC194 | Vila, Silvia; Badosa, Esther; Montesinos, Emilio; Feliu, Lidia; Planas, Marta | European Journal of Organic Chemistry | 2015 | | 15 |
| cpdart0064 | Synthesis and Preliminary Evaluation of Novel Bone-targeting NSAIDs Prodrugs based on Glutamic Acid Oligopeptides | Zhao, Yi; He, Dongsheng; Ma, Lifang; Guo, Li | Letters in Drug Design & Discovery | 2015 | | 12 |
| cpdart0065 | Synthesis and mass spectrometry analysis of quaternary cryptando-peptidic conjugates | Bachor, Remigiusz; Kluczyk, Alicja; Stefanowicz, Piotr; Szewczuk, Zbigniew | Journal of Peptide Science | 2015 | | 3 |
| cpdart0066 | Propargyloxyproline regio- and stereoisomers for Click-conjugation of peptides: Synthesis and application in linear and cyclic peptides | Northfield, Susan E.; Mountford, Simon J.; Wielens, Jerome; Liu, Mengjie; Zhang, Lei; Herzog, Herbert; Holliday, Nicholas D.; Scanlon, Martin J.; Parker, Michael W.; Chalmers, David K.; Thompson, Philip E. | Australian Journal of Chemistry | 2015 | | 25 |
| cpdart0067 | Ligation of anti-cancer drugs to self-assembling ultrashort peptides by click chemistry for localized therapy | Reithofer, Michael R.; Chan, Kiat-Hwa; Lakshmanan, Anupama; Lam, Dang Hoang; Mishra, Archana; Gopalan, Began; Joshi, Mangesh; Wang, Shu; Hauser, Charlotte A. E. | Chemical Science | 2014 | | 4 |
| cpdart0068 | Targeted Delivery of Ubiquitin-Conjugated BH3 Peptide-Based Mcl-1 Inhibitors into Cancer Cells | Muppidi, Avinash; Doi, Kenichiro; Edwardraja, Selvakumar; Pulavarti, Surya V. S. R. K.; Szyperski, Thomas; Wang, Hong-Gang; Lin, Qing | Bioconjugate Chemistry | 2014 | | 1 |
| cpdart0069 | Enthalpy-driven nuclease-like activity and mechanism of peptide-chlorambucil conjugates | Yang, Robin C. K.; Huang, Jonathan T. B.; Chen, Yu-Ling; Hung, Chia-Chun; Liao, Mokai; Yao, Wen-Chen; Chen, Chiu-Heng; Liou, Chien-Chung; Waring, Michael J.; Sheh, Leung | Organic & Biomolecular Chemistry | 2014 | | 2 |
| cpdart0070 | Macrolide-Peptide Conjugates as Probes of the Path of Travel of the Nascent Peptides through the Ribosome | Washington, Arren Z.; Benicewicz, Derek B.; Canzoneri, Joshua C.; Fagan, Crystal E.; Mwakwari, Sandra C.; Maehigashi, Tatsuya; Dunham, Christine M.; Oyelere, Adegboyega K. | ACS Chemical Biology | 2014 | | 8 |
| cpdart0071 | C60 Pyrrolidine Bis-carboxylic Acid Derivative as a Versatile Precursor for Biocompatible Fullerenes | Aroua, Safwan; Schweizer, W. Bernd; Yamakoshi, Yoko | Organic Letters | 2014 | | 3 |
| cpdart0072 | Chromatography- and Lyophilization-Free Synthesis of a Peptide-Linker Conjugate | Magano, Javier; Bock, Brandon; Brennan, John; Farrand, Douglas; Lovdahl, Michael; Maloney, Mark T.; Nadkarni, Durgesh; Oliver, Wendy K.; Pozzo, Mark J.; Teixeira, John J.; Wang, Jian; Rizzo, John; Tumelty, David | Organic Process Research & Development | 2014 | | 1 |
| cpdart0073 | Shuttle-Cargo Fusion Molecules of Transport Peptides and the hD2/3 Receptor Antagonist Fallypride: A Feasible Approach To Preserve Ligand-Receptor Binding? | Wangler, Carmen; Chowdhury, Shafinaz; Hofner, Georg; Djurova, Petia; Purisima, Enrico O.; Bartenstein, Peter; Wangler, Bjorn; Fricker, Gert; Wanner, Klaus T.; Schirrmacher, Ralf | Journal of Medicinal Chemistry | 2014 | | 46 |
| cpdart0074 | Design, synthesis, and evaluation of derivatives of the fat-accumulation inhibitor ternatin: toward ternatin molecular probes | Kawazoe, Yoshinori; Tanaka, Yoko; Omura, Sachikazu; Uemura, Daisuke | Tetrahedron Letters | 2014 | | 16 |
| cpdart0075 | Bisubstrate UDP-peptide conjugates as human O-GlcNAc transferase inhibitors | Borodkin, Vladimir S.; Schimpl, Marianne; Gundogdu, Mehmet; Rafie, Karim; Dorfmueller, Helge C.; Robinson, David A.; van Aalten, Daan M. F. | Biochemical Journal | 2014 | | 2 |
| cpdart0076 | Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery System | Barile, Elisa; Wang, Si; Das, Swadesh K.; Noberini, Roberta; Dahl, Russell; Stebbins, John L.; Pasquale, Elena B.; Fisher, Paul B.; Pellecchia, Maurizio | ChemMedChem | 2014 | | 4 |
| cpdart0077 | Synthesis, Spectroscopic, and Photophysical Characterization and Photosensitizing Activity toward Prokaryotic and Eukaryotic Cells of Porphyrin-Magainin and -Buforin Conjugates | Dosselli, Ryan; Ruiz-Gonzalez, Ruben; Moret, Francesca; Agnolon, Valentina; Compagnin, Chiara; Mognato, Maddalena; Sella, Valentina; Agut, Montserrat; Nonell, Santi; Gobbo, Marina; Reddi, Elena | Journal of Medicinal Chemistry | 2014 | | 5 |
| cpdart0078 | Design, Synthesis, and Biological Evaluation of Highly Potent Small Molecule-Peptide Conjugates as New HIV-1 Fusion Inhibitors | Wang, Chao; Shi, Weiguo; Cai, Lifeng; Lu, Lu; Wang, Qian; Zhang, Tianhong; Li, Jinglai; Zhang, Zhenqing; Wang, Kun; Xu, Liang; Jiang, Xifeng; Jiang, Shibo; Liu, Keliang | Journal of Medicinal Chemistry | 2013 | | 4 |
| cpdart0079 | Synthesis, enzymatic stability and in vitro cytostatic effect of Daunorubicin-GnRH-III derivative dimers | Schreier, Verena Natalie; Mezo, Gabor; Orban, Erika; Duerr, Claudia; Marquardt, Andreas; Manea, Marilena | Bioorganic & Medicinal Chemistry Letters | 2013 | | 6 |
| cpdart0080 | Thiazolidinone-Peptide Hybrids as Dengue Virus Protease Inhibitors with Antiviral Activity in Cell Culture | Nitsche, Christoph; Schreier, Verena N.; Behnam, Mira A. M.; Kumar, Anil; Bartenschlager, Ralf; Klein, Christian D. | Journal of Medicinal Chemistry | 2013 | | 60 |
| cpdart0081 | Phthalocyanine-Peptide Conjugates: Receptor-Targeting Bifunctional Agents for Imaging and Photodynamic Therapy | Ranyuk, Elena; Cauchon, Nicole; Klarskov, Klaus; Guerin, Brigitte; van Lier, Johan E. | Journal of Medicinal Chemistry | 2013 | | 5 |
| cpdart0082 | Cellular uptake and cytotoxicity of drug-peptide conjugates regulated by conjugation site | Zhang, Pengcheng; Cheetham, Andrew G.; Lock, Lye Lin; Cui, Honggang | Bioconjugate Chemistry | 2013 | | 6 |
| cpdart0083 | Synthesis and Antimalarial Bioassay of Quinine - Peptide Conjugates | Panda, Siva S.; Ibrahim, Mohamed A.; Kuecuekbay, Hasan; Meyers, Marvin J.; Sverdrup, Francis M.; El-Feky, Said A.; Katritzky, Alan R. | Chemical Biology & Drug Design | 2013 | | 4 |
| cpdart0084 | Cholesterol-peptide hybrids to form liposome-like vesicles for gene delivery | Tang, Qiong; Cao, Bin; Wu, Haiyan; Cheng, Gang | PLoS One | 2013 | | 4 |
| cpdart0085 | Cell-Penetrating Bisubstrate-Based Protein Kinase C Inhibitors | van Wandelen, Loek T. M.; van Ameijde, Jeroen; Ismail-Ali, Ahmed F.; van Ufford, H. C. Quarles; Vijftigschild, Lodewijk A. W.; Beekman, Jeffrey M.; Martin, Nathaniel I.; Ruijtenbeek, Rob; Liskamp, Rob M. J. | ACS Chemical Biology | 2013 | | 3 |
| cpdart0086 | Betulonic acid-peptide conjugates: synthesis and evaluation of anti-inflammatory activity | Govdi, Anastasiya I.; Vasilevsky, Sergei F.; Sokolova, Nadezhda V.; Sorokina, Irina V.; Tolstikova, Tatyana G.; Nenajdenko, Valentine G. | Mendeleev Communications | 2013 | | 6 |
| cpdart0087 | Peptide conjugates of 4-aminocyclophosphamide as prodrugs of phosphoramide mustard for selective activation by prostate-specific antigen (PSA) | Jiang, Yongying; Hu, Longqin | Bioorganic & Medicinal Chemistry | 2013 | | 8 |
| cpdart0088 | Novel water-soluble prodrugs of acyclovir cleavable by the dipeptidyl-peptidase IV (DPP IV/CD26) enzyme | Diez-Torrubia, Alberto; Cabrera, Silvia; de Castro, Sonia; Garcia-Aparicio, Carlos; Mulder, Gwenn; De Meester, Ingrid; Camarasa, Maria-Jose; Balzarini, Jan; Velazquez, Sonsoles | European Journal of Medicinal Chemistry | 2013 | | 8 |
| cpdart0089 | Organogels of triterpenoid-tripeptide conjugates: Encapsulation of dye molecules and basicity increase associated with aggregation | Lu, Jinrong; Gao, Yuxia; Wu, Jindan; Ju, Yong | RSC Advances | 2013 | | 2 |
| cpdart0090 | Peptide-Drug Conjugate Linked via a Disulfide Bond for Kidney Targeted Drug Delivery | Geng, Qian; Sun, Xun; Gong, Tao; Zhang, Zhi-Rong | Bioconjugate Chemistry | 2012 | | 2 |
| cpdart0091 | The First Generation of β‐Galactosidase‐Responsive Prodrugs Designed for the Selective Treatment of Solid Tumors in Prodrug Monotherapy | Legigan, Thibaut; Clarhaut, Jonathan; Tranoy-Opalinski, Isabelle; Monvoisin, Arnaud; Renoux, Brigitte; Thomas, Mikael; Le Pape, Alain; Lerondel, Stephanie; Papot, Sebastien | Angewandte Chemie, International Edition | 2012 | | 2 |
| cpdart0092 | Cell-penetrating γ-peptide/antimicrobial undecapeptide conjugates with anticancer activity | Roses, Cristina; Carbajo, Daniel; Sanclimens, Gloria; Farrera-Sinfreu, Josep; Blancafort, Adriana; Oliveras, Gloria; Cirac, Anna D.; Bardaji, Eduard; Puig, Teresa; Planas, Marta; Feliu, Lidia; Albericio, Fernando; Royo, Miriam | Tetrahedron | 2012 | | 2 |
| cpdart0093 | Modular synthesis of supramolecular ureidopyrimidinone-peptide conjugates using an oxime ligation strategy | Kieltyka, Roxanne E.; Bastings, Maartje M. C.; van Almen, Geert C.; Besenius, Pol; Kemps, Erwin W. L.; Dankers, Patricia Y. W. | Chemical Communications | 2012 | | 7 |
| cpdart0094 | Optimization of BACE1 inhibition of tripartite structures by modification of membrane anchors, spacers and pharmacophores - development of potential agents for the treatment of Alzheimer's disease | Linning, Philipp; Haussmann, Ute; Beyer, Isaak; Weidlich, Sebastian; Schieb, Heinke; Wiltfang, Jens; Klafki, Hans-Wolfgang; Knoelker, Hans-Joachim | Organic & Biomolecular Chemistry | 2012 | | 17 |
| cpdart0095 | A general route to xyloglucan-peptide conjugates for the activation of cellulose surfaces | Araujo, Ana Catarina; Nakhai, Azadeh; Ruda, Marcus; Slaettegard, Rikard; Gatenholm, Paul; Brumer, Harry | Carbohydrate Research | 2012 | | 3 |
| cpdart0096 | Synthesis of [12]aneN3-dipeptide conjugates as metal-free DNA nucleases | Li, Zhi-Fen; Chen, Hua-Long; Zhang, Li-Jun; Lu, Zhong-Lin | Bioorganic & Medicinal Chemistry Letters | 2012 | | 8 |
| cpdart0097 | DOTA-tris(OPp ester) as a bifunctional prochelator for the preparation of DOTA-peptide conjugates | Jamous, Mazen; Haberkorn, Uwe; Mier, Walter | Tetrahedron Letters | 2012 | | 3 |
| cpdart0098 | Efficient formation of heterodimers from peptides and proteins using unsymmetrical polyfluorophenyl esters of dicarboxylic acids | Slosarczyk, Adam T.; Baltzer, Lars | Journal of Peptide Science | 2012 | | 8 |
| cpdart0099 | Synthesis of small molecule-peptide conjugates as potential whitening agents | Lee, Hye-Suk; Shin, Kyong-Hoon; Ryu, Geun-Seok; Chi, Gyeong-Yup; Cho, In-Shik; Kim, Han-Young | Bulletin of the Korean Chemical Society | 2012 | | 18 |
| cpdart0100 | Enhancing cellular uptake of activable cell-penetrating peptide-doxorubicin conjugate by enzymatic cleavage | Shi, Nian-Qiu; Gao, Wei; Xiang, Bai; Qi, Xian-Rong | International Journal of Nanomedicine | 2012 | | 1 |
| cpdart0101 | β-Lactam-host defence peptide conjugates as antibioticprodrug candidates targeting resistant bacteria | Desgranges, Stephane; Ruddle, Carol C.; Burke, Liam P.; McFadden, Tara M.; O'Brien, John E.; Fitzgerald-Hughes, Deirdre; Humphreys, Hilary; Smyth, Timothy P.; Devocelle, Marc | RSC Advances | 2012 | | 3 |
| cpdart0102 | Enhanced Cellular Uptake of a New, in Silico Identified Antitubercular Candidate by Peptide Conjugation | Horvati, Kata; Bacsa, Bernadett; Szabo, Nora; David, Sandor; Mezo, Gabor; Grolmusz, Vince; Vertessy, Beata; Hudecz, Ferenc; Bosze, Szilvia | Bioconjugate Chemistry | 2012 | | 2 |
| cpdart0103 | Methotrexate-cIBR conjugate for targeting methotrexate to leukocytes: Conjugate stability and in vivo efficacy in suppressing rheumatoid arthritis | Majumdar, Sumit; Anderson, Meagan E.; Xu, Christine R.; Yakovleva, Tatyana V.; Gu, Leo C.; Malefyt, Thomas R.; Siahaan, Teruna J. | Journal of Pharmaceutical Sciences | 2012 | | 7 |
| cpdart0104 | A New Family of Highly Potent Inhibitors of Microbes: Synthesis and Conjugation of Elastin Based Peptides to Piperazine Derivative | Suhas, R.; Chandrashekar, S.; Gowda, D. Channe | International Journal of Peptide Research and Therapeutics | 2012 | | 14 |
| cpdart0105 | Lipopolysaccharide Neutralizing Peptide-Porphyrin Conjugates for Effective Photoinactivation and Intracellular Imaging of Gram-Negative Bacteria Strains | Liu, Fang; Soh Yan Ni, Annie; Lim, Yingjie; Mohanram, Harini; Bhattacharjya, S.; Xing, Bengang | Bioconjugate Chemistry | 2012 | | 1 |
| cpdart0106 | Microwave-assisted formation of peptide-vitamin conjugates | El-Nachef, Claudia; Bajaj, Kiran; Koblick, Jacqueline; Katritzky, Alan R. | European Journal of Organic Chemistry | 2012 | | 11 |
| cpdart0107 | Synthesis of peptide conjugates of mestranol by a 1,3-dipolar cycloaddition click reaction | Sokolova, N. V.; Nenajdenko, V. G. | Chemistry of Heterocyclic Compounds | 2012 | | 6 |
| cpdart0108 | Synthesis of α-Trifluoromethyl-α-hydroxy Acid-Peptide Conjugates via Click Chemistry | Sokolova, Nadezhda V.; Vorobyeva, Daria V.; Osipov, Sergey N.; Vasilyeva, Tamara P.; Nenajdenko, Valentine G. | Synthesis | 2012 | | 14 |
| cpdart0109 | Syntheses of chiral N-(protected) tri- and tetrapeptide conjugates | Bajaj, Kiran; Panda, Siva S.; El-Nachef, Claudia; Katritzky, Alan R. | Chemical Biology & Drug Design | 2012 | | 7 |
| cpdart0110 | Novel cinnamic acid/4-aminoquinoline conjugates bearing non-proteinogenic amino acids: Towards the development of potential dual action antimalarials | Perez, Bianca C.; Teixeira, Catia; Figueiras, Marta; Gut, Jiri; Rosenthal, Philip J.; Gomes, Jose R. B.; Gomes, Paula | European Journal of Medicinal Chemistry | 2012 | | 17 |
| cpdart0112 | Biological Evaluation of a Novel Doxorubicin-Peptide Conjugate for Targeted Delivery to EGF Receptor-Overexpressing Tumor Cells | Ai, Shibin; Duan, Jianli; Liu, Xin; Bock, Stephanie; Tian, Yuan; Huang, Zebo | Molecular Pharmaceutics | 2011 | | 2 |
| cpdart0113 | A New Daunomycin-Peptide Conjugate: Synthesis, Characterization and the Effect on the Protein Expression Profile of HL-60 Cells in Vitro | Orban, Erika; Manea, Marilena; Marquadt, Andreas; Banoczi, Zoltan; Csik, Gabriella; Fellinger, Erzsebet; Bosze, Szilvia; Hudecz, Ferenc | Bioconjugate Chemistry | 2011 | | 1 |
| cpdart0114 | Synthesis of elastin based peptides conjugated to benzisoxazole as a new class of potent antimicrobials - A novel approach to enhance biocompatibility | Suhas, R.; Chandrashekar, S.; Gowda, D. Channe | European Journal of Medicinal Chemistry | 2011 | | 14 |
| cpdart0115 | New pemetrexed-peptide conjugates: synthesis, characterization and in vitro cytostatic effect on non-small cell lung carcinoma (NCI-H358) and human leukemia (HL-60) cells | Miklan, Zsanett; Orban, Erika; Banoczi, Zoltan; Hudecz, Ferenc | Journal of Peptide Science | 2011 | | 6 |
| cpdart0116 | Synthesis and antibacterial activity of amphiphilic lysine-ligated neomycin B conjugates | Bera, Smritilekha; Zhanel, George G.; Schweizer, Frank | Carbohydrate Research | 2011 | | 1 |
| cpdart0117 | Synthesis and Self-Assembly of Oligo(p-phenylenevinylene) Peptide Conjugates in Water | Mba, Miriam; Moretto, Alessandro; Armelao, Lidia; Crisma, Marco; Toniolo, Claudio; Maggini, Michele | Chemistry - A European Journal | 2011 | | 2 |
| cpdart0118 | Novel β-carboline-tripeptide conjugates attenuate mesenteric ischemia/reperfusion injury in the rat | Bi, Wei; Bi, Yue; Xue, Ping; Zhang, Yanrong; Gao, Xiang; Wang, Zhibo; Li, Meng; Baudy-Floc'h, Michele; Ngerebara, Nathaniel; Li, Xiaoxu; Gibson, K. Michael; Bi, Lanrong | European Journal of Medicinal Chemistry | 2011 | | 36 |
| cpdart0119 | A new class of β-carboline alkaloid-peptide conjugates with therapeutic efficacy in acute limb ischemia/reperfusion injury | Bi, Wei; Bi, Yue; Xue, Ping; Zhang, Yanrong; Gao, Xiang; Wang, Zhibo; Li, Meng; Baudy-Floc'h, Michele; Ngerebara, Nathaniel; Michael Gibson, K.; Bi, Lanrong | European Journal of Medicinal Chemistry | 2011 | | 26 |
| cpdart0120 | Syntheses and DNA binding of new cationic porphyrin-tetrapeptide conjugates | Mezo, Gabor; Herenyi, Levente; Habdas, Jan; Majer, Zsuzsa; Mysliwa-Kurdziel, Beata; Toth, Katalin; Csik, Gabriella | Biophysical Chemistry | 2011 | | 2 |
| cpdart0121 | Solid phase synthesis and biological activity of tuftsin conjugates | Kukowska-Kaszuba, Magdalena; Dzierzbicka, Krystyna; Serocki, Marcin; Skladanowski, Andrzej | Journal of Medicinal Chemistry | 2011 | | 34 |
| cpdart0123 | Synthesis and optimization of hyaluronic acid-methotrexate conjugates to maximize benefit in the treatment of osteoarthritis | Homma, Akie; Sato, Haruhiko; Tamura, Tatsuya; Okamachi, Akira; Emura, Takashi; Ishizawa, Takenori; Kato, Tatsuya; Matsuura, Tetsu; Sato, Shigeo; Higuchi, Yoshinobu; Watanabe, Tomoyuki; Kitamura, Hidetomo; Asanuma, Kentaro; Yamazaki, Tadao; Ikemi, Masahisa; Kitagawa, Hironoshin; Morikawa, Tadashi; Ikeya, Hitoshi; Maeda, Kazuaki; Takahashi, Koichi; Nohmi, Kenji; Izutani, Noriyuki; Kanda, Makoto; Suzuki, Ryohchi | Bioorganic & Medicinal Chemistry | 2010 | | 27 |
| cpdart0124 | Synthesis and in Vitro Antitumor Effect of Vinblastine Derivative-Oligoarginine Conjugates | Banoczi, Zoltan; Gorka-Kereskenyi, Almos; Remenyi, Judit; Orban, Erika; Hazai, Laszlo; Tokesi, Natalia; Olah, Judit; Ovadi, Judit; Beni, Zoltan; Hada, Viktor; Szantay, Csaba Jr.; Hudecz, Ferenc; Kalaus, Gyorgy; Szantay, Csaba | Bioconjugate Chemistry | 2010 | | 6 |
| cpdart0125 | Application of the Dipeptidyl Peptidase IV (DPPIV/CD26) Based Prodrug Approach to Different Amine-Containing Drugs | Diez-Torrubia, Alberto; Garcia-Aparicio, Carlos; Cabrera, Silvia; De Meester, Ingrid; Balzarini, Jan; Camarasa, Maria-Jose; Velazquez, Sonsoles | Journal of Medicinal Chemistry | 2010 | | 16 |
| cpdart0126 | Evaluation of amphiphilic aminoglycoside-peptide triazole conjugates as antibacterial agents | Bera, Smritilekha; Zhanel, George G.; Schweizer, Frank | Bioorganic & Medicinal Chemistry | 2010 | | 13 |
| cpdart0127 | Synthesis of DOTA-Conjugated Multimeric [Tyr3]Octreotide Peptides via a Combination of Cu(I)-Catalyzed "Click"" Cycloaddition and Thio Acid/Sulfonyl Azide ""Sulfo-Click"" Amidation and Their in Vivo Evaluation" | Yim, Cheng-Bin; Dijkgraaf, Ingrid; Merkx, Remco; Versluis, Cees; Eek, Annemarie; Mulder, Gwenn E.; Rijkers, Dirk T. S.; Boerman, Otto C.; Liskamp, Rob M. J. | Journal of Medicinal Chemistry | 2010 | | 4 |
| cpdart0128 | Synthesis of Mono-ADP-Ribosylated Oligopeptides Using Ribosylated Amino Acid Building Blocks | van der Heden van Noort, Gerbrand J.; van der Horst, Maarten G.; Overkleeft, Herman S.; van der Marel, Gijsbert A.; Filippov, Dmitri V. | Journal of the American Chemical Society | 2010 | | 5 |
| cpdart0129 | Structural Design, Solid‐Phase Synthesis and Activity of Membrane‐Anchored β‐Secretase Inhibitors on Aβ Generation from Wild‐Type and Swedish‐Mutant APP | Schieb, Heinke; Weidlich, Sebastian; Schlechtingen, Georg; Linning, Philipp; Jennings, Gary; Gruner, Margit; Wiltfang, Jens; Klafki, Hans-Wolfgang; Knoelker, Hans-Joachim | Chemistry - A European Journal | 2010 | | 9 |
| cpdart0131 | Biological evaluation of paclitaxel-peptide conjugates as a model for MMP2-targeted drug delivery | Yamada, Roppei; Kostova, Maya B.; Anchoori, Ravi Kumar; Xu, Shili; Neamati, Nouri; Khan, Saeed R. | Cancer Biology & Therapy | 2010 | | 3 |
| cpdart0132 | "Click" synthesis of small molecule-peptide conjugates for organelle-specific delivery and inhibition of lysosomal cysteine proteases" | Loh, Yuhui; Shi, Haibin; Hu, Mingyu; Yao, Shao Q. | Chemical Communications | 2010 | | 3 |
| cpdart0133 | A DOTA-peptide conjugate by copper-free click chemistry | Martin, Molly E.; Parameswarappa, Sharavathi G.; O'Dorisio, M. Sue; Pigge, F. Christopher; Schultz, Michael K. | Bioorganic & Medicinal Chemistry | 2010 | | 2 |
| cpdart0134 | Facile synthesis of peptide-porphyrin conjugates: Towards artificial catalase | Umezawa, Naoki; Matsumoto, Nobuyoshi; Iwama, Shinsuke; Kato, Nobuki; Higuchi, Tsunehiko | Bioorganic & Medicinal Chemistry | 2010 | | 1 |
| cpdart0135 | Influence of the number and distribution of NLS peptides on the photosensitizing activity of multimeric porphyrin-NLS | Sibrian-Vazquez, Martha; Jensen, Timothy J.; Vicente, M. Graca H. | Organic & Biomolecular Chemistry | 2010 | | 3 |
| cpdart0136 | A Metal-Free DNA Nuclease Based on a Cyclic Peptide Scaffold | Alkhader, Shadad; Ezra, Aviva; Kasparkova, Jana; Brabec, Viktor; Yavin, Eylon | Bioconjugate Chemistry | 2010 | | 18 |
| cpdart0137 | Synthesis and Characterization of New Galanthamine Derivatives Comprising Peptide Moiety | Lyubomir T. Vezenkov, Maria G. Georgieva, Dantcho L. Danalev, Tchavdar B. Ivanov, Galya I. Ivanova | Protein & Peptide Letters | 2009 | | 7 |
| cpdart0138 | Novel type 1 photosensitizers: viability of leukemia cells exposed to reactive intermediates generated in situ by in vitro photofragmentation | Raghavan Rajagopalan, Amol Karwa, Przemyslaw M. Lusiak, Kripa Srivastava, Amruta R. Poreddy, Raghootama S. Pandurangi, Karen P. Galen, William L. Neumann, Gary E. Cantrell, Richard B. Dorshow | Proc. SPIE 7380, Photodynamic Therapy: Back to the Future | 2009 | | 1 |
| cpdart0139 | New daunomycin–oligoarginine conjugates: Synthesis, characterization, and effect on human leukemia and human hepatoma cells | Zsanett Miklán; Erika Orbán; Gabriella Csík; Gitta Schlosser; Anna Magyar; Ferenc Hudecz | Peptide Science | 2009 | | 6 |
| cpdart0140 | Design and synthesis of novel histone deacetylase inhibitor derived from nuclear localization signal peptide | Joshua C.Canzoneri; Po C.Chen; Adegboyega K.Oyelere | Bioorganic & Medicinal Chemistry Letters | 2009 | | 6 |
| cpdart0141 | A novel L-ascorbic acid and peptide conjugate with increased stability and collagen biosynthesis | Ho-Il Choi, Jong-Il Park, Heung-Jae Kim, Dong-Won Kim, Soung-Soo Kim | BMB Reports | 2009 | | 1 |
| cpdart0142 | Peptide Targeting of Platinum Anti-Cancer Drugs | Ndinguri, Margaret W.; Solipuram, Rajasree; Gambrell, Robert P.; Aggarwal, Sita; Hammer, Robert P. | Bioconjugate Chemistry | 2009 | | 2 |
| cpdart0143 | Towards the conformational mimicry of the measles virus HNE loop: design, synthesis and biological evaluation of a cyclic bile acid-peptide conjugate | Bode, Catherine A.; Bechet, Tom; Prodhomme, Emmanuel; Gheysen, Katelijne; Gregoir, Pieter; Martins, Jose C.; Muller, Claude P.; Madder, Annemieke | Organic & Biomolecular Chemistry | 2009 | | 8 |
| cpdart0144 | An efficient route to VEGF-like peptide porphyrin conjugates via microwave-assisted 'click-chemistry' | Bakleh, M. E.; Sol, V.; Estieu-Gionnet, K.; Granet, R.; Deleris, G.; Krausz, P. | Tetrahedron | 2009 | | 2 |
| cpdart0145 | Synthesis and preliminary evaluation in vitro of novel naproxen-dendritic peptide conjugates | Ouyang, Liang; Zhang, Jing; Pan, Junzhu; Yan, Linna; Guo, Li | Drug Delivery | 2009 | | 7 |
| cpdart0146 | An improved synthesis of releasable luciferin-CPP conjugates | Eiriksdottir, Emelia; Langel, Uelo; Rosenthal-Aizman, Katri | Tetrahedron Letters | 2009 | | 3 |
| cpdart0147 | Silver-Catalyzed azaGly Ligation. Application to the Synthesis of Azapeptides and of Lipid-Peptide Conjugates | Ollivier, Nathalie; Besret, Soizic; Blanpain, Annick; Melnyk, Oleg | Bioconjugate Chemistry | 2009 | | 3 |
| cpdart0148 | Novel hyaluronic acid-methotrexate conjugates for osteoarthritis treatment | Homma, Akie; Sato, Haruhiko; Okamachi, Akira; Emura, Takashi; Ishizawa, Takenori; Kato, Tatsuya; Matsuura, Tetsu; Sato, Shigeo; Tamura, Tatsuya; Higuchi, Yoshinobu; Watanabe, Tomoyuki; Kitamura, Hidetomo; Asanuma, Kentaro; Yamazaki, Tadao; Ikemi, Masahisa; Kitagawa, Hironoshin; Morikawa, Tadashi; Ikeya, Hitoshi; Maeda, Kazuaki; Takahashi, Koichi; Nohmi, Kenji; Izutani, Noriyuki; Kanda, Makoto; Suzuki, Ryochi | Bioorganic & Medicinal Chemistry | 2009 | | 4 |
| cpdart0149 | Estrano[17,16-e]pyrimidine-amino acid and estrano[17,16-e]pyrimidine-peptide conjugates | Matsumoto, Tomohiro; Shiine, Kodai; Mataka, Shuntaro; Thiemann, Thies | Journal of Chemical Research | 2009 | | 7 |
| cpdart0150 | A new water soluble 3,6,9-trioxaundecanedioic acid-based linker and biotinylating reagent | Bartos, Adam; Hudecz, Ferenc; Uray, Katalin | Tetrahedron Letters | 2009 | | 3 |
| cpdart0151 | Dipole effects on molecular and electronic structures in a novel conjugate of oligo(phenyleneethynylene) and helical peptide | Nakayama, Hidenori; Morita, Tomoyuki; Kimura, Shunsaku | Physical Chemistry Chemical Physics | 2009 | | 2 |
| cpdart0152 | 3D QSAR of novel estrogen-RGD peptide conjugates: Getting insight into structural dependence of anti-osteoporosis activity and side effect of estrogen in ERT | Zhao, Ming; Liu, Jiangyuan; Zhang, Xiaoyi; Peng, Li; Li, Chunyu; Peng, Shiqi | Bioorganic & Medicinal Chemistry | 2009 | | 17 |
| cpdart0153 | Synthesis and stereochemical preference of peptide 4-aminocyclophosphamide conjugates as potential prodrugs of phosphoramide mustard for activation by prostate-specific antigen (PSA) | Jiang, Yongying; Di Paola, Robert S.; Hu, Longqin | Bioorganic & Medicinal Chemistry | 2009 | | 4 |
| cpdart0154 | Synthesis, evaluation and 3D QSAR analysis of novel estradiol-RGD octapeptide conjugates with oral anti-osteoporosis activity | Liu, Jiangyuan; Zhang, Xiaoyi; Zhao, Ming; Peng, Shiqi | European Journal of Medicinal | 2009 | | 16 |
| cpdart0155 | Effect of Modification of the Physicochemical Properties of ICAM-1-Derived Peptides on Internalization and Intracellular Distribution in the Human Leukemic Cell Line HL-60 | Majumdar, Sumit; Tejo, Bimo A.; Badawi, Ahmed H.; Moore, David; Krise, Jeffrey P.; Siahaan, Teruna J. | Molecular Pharmaceutics | 2009 | | 2 |
| cpdart0156 | Design and efficient synthesis of novel ascorbyl conjugated peptide with high collagen biosynthesis stimulating effects | Choi, Ho-Il; Kim, Heung-Jae; Park, Jong-Il; Shin, Eun-Ho; Kim, Dong-Won; Kim, Soung-Soo | Bioorganic & Medicinal Chemistry Letters | 2009 | | 2 |
| cpdart0157 | Synthesis and anti-cancer activity of covalent conjugates of artemisinin and a transferrin-receptor targeting peptide | Oh, Steve; Kim, Byung Ju; Singh, Narendra P.; Lai, Henry; Sasaki, Tomikazu | Cancer Letters | 2009 | | 2 |
| cpdart0158 | Synthesis and Biological Evaluation of Vinca Alkaloids and Phomopsin Hybrids | Ngo, Quoc Anh; Roussi, Fanny; Cormier, Anthony; Thoret, Sylviane; Knossow, Marcel; Guenard, Daniel; Gueritte, Francoise | Journal of Medicinal Chemistry | 2009 | | 5 |
| cpdart0159 | Triple Hybrids of Steroids, Spiroketals, and Oligopeptides as New Biomolecular Chimeras | Banerjee, Abhisek; Sergienko, Eduard; Vasile, Stefan; Gupta, Vineet; Vuori, Kristiina; Wipf, Peter | Organic Letters | 2009 | | 10 |
| cpdart0160 | Synthesis of daunomycin-oligoarginine conjugates and their effect on human leukemia cells (HL-60) | Banoczi, Zoltan; Peregi, Balazs; Orban, Erika; Szabo, Rita; Hudecz, Ferenc | ARKIVOC | 2008 | | 3 |
| cpdart0161 | Oligo(p-phenylenevinylene)-Peptide Conjugates: Synthesis and Self-Assembly in Solution and at the Solid-Liquid Interface | Matmour, Rachid; De Cat, Inge; George, Subi J.; Adriaens, Wencke; Leclere, Philippe; Bomans, Paul H. H.; Sommerdijk, Nico A. J. M.; Gielen, Jeroen C.; Christianen, Peter C. M.; Heldens, Jeroen T.; van Hest, Jan C. M.; Loewik, Dennis W. P. M.; De Feyter, Steven; Meijer, E. W.; Schenning, Albertus P. H. J. | Journal of the American Chemical Society | 2008 | | 1 |
| cpdart0162 | Photoinduced Cytotoxicity and Biodistribution of Prostate Cancer Cell-Targeted Porphyrins | Sehgal, Inder; Sibrian-Vazquez, Martha; Vicente, M. Graca H. | Journal of Medicinal Chemistry | 2008 | | 2 |
| cpdart0163 | In vitro and in vivo evaluation of doxorubicin conjugates with the divalent peptide E-[c(RGDfK)2] that targets integrin αvβ3 | Ryppa, Claudia; Mann-Steinberg, Hagit; Fichtner, Iduna; Weber, Holger; Satchi-Fainaro, Ronit; Biniossek, Martin L.; Kratz, Felix | Bioconjugate Chemistry | 2008 | | 1 |
| cpdart0164 | A cell-penetrating peptidic GRP78 ligand for tumor cell-specific prodrug therapy | Yoneda, Yoshiyuki; Steiniger, Sebastian C. J.; Capkova, Katerina; Mee, Jenny M.; Liu, Ying; Kaufmann, Gunnar F.; Janda, Kim D. | Bioorganic & Medicinal Chemistry Letters | 2008 | | 2 |
| cpdart0165 | 1-Ethoxyethylidene, a New Group for the Stepwise SPPS of Aminooxyacetic Acid Containing Peptides | Foillard, Stephanie; Ohsten Rasmussen, Martin; Razkin, Jesus; Boturyn, Didier; Dumy, Pascal | Journal of Organic Chemistry | 2008 | | 3 |
| cpdart0166 | Syntheses and cellular studies of water soluble porphyrin-peptide conjugates | Sibrian-Vazquez, Martha; Jensen, Timothy J.; Hammer, Robert P.; Vicente, M. Graca H. | Proceedings of SPIE-The International Society for Optical Engineering | 2008 | | 6 |
| cpdart0167 | Synthesis of a coumarin-histone conjugate for HAT fluorescent assay | Chen, Ziyue; Zheng, Yujun George | Heterocyclic Communications | 2008 | | 1 |
| cpdart0168 | Reversible switching of substrate activity of poly-N-isopropylacrylamide peptide conjugates | Molawi, Kian; Studer, Armido | Chemical Communications | 2007 | | 7 |
| cpdart0169 | Efficient conversion of tetrapeptide-based TSAO prodrugs to the parent drug by dipeptidyl-peptidase IV (DPPIV/CD26) | Garcia-Aparicio, Carlos; Diez-Torrubia, Alberto; Balzarini, Jan; Lambeir, Anne-Marie; Velazquez, Sonsoles; Camarasa, Maria-Jose | Antiviral Research | 2007 | | 8 |
| cpdart0170 | Design and synthesis of paclitaxel conjugated with an ErbB2-recognizing peptide, EC-1 | Li, Peng; Jiang, Sheng; Pero, Stephanie C.; Oligino, Lyn; Krag, David N.; Michejda, Christopher J.; Roller, Peter P. | Biopolymers | 2007 | | 2 |
| cpdart0171 | Validation of a solid-phase-bound steroid scaffold for the synthesis of novel cyclic peptidosteroids | Bode, Catherine A.; Muller, Claude P.; Madder, Annemieke | Journal of Peptide Science | 2007 | | 6 |
| cpdart0172 | Biosynthetic Tailoring of Microcin E492m: Post-translational Modification Affords an Antibacterial Siderophore-Peptide Conjugate | Nolan, Elizabeth M.; Fischbach, Michael A.; Koglin, Alexander; Walsh, Christopher T. | Journal of the American Chemical Society | 2007 | | 3 |
| cpdart0173 | Synthesis and antitumor activity of peptide-paclitaxel conjugates | Papas, Serafim; Akoumianaki, Tonia; Kalogiros, Christos; Hadjiarapoglou, Lazaros; Theodoropoulos, Panayiotis A.; Tsikaris, Vassilios | Journal of Peptide Science | 2007 | | 3 |
| cpdart0174 | Synthesis and assessment of a novel peptide conjugate to deliver phenytoin for wound repair | Kennedy, C. A.; Chan, F. C.; DeVocelle, M.; Meaney, C.; Bouchier-Hayes, D. J.; Kelly, J. G. | Journal of Drug Delivery Science and Technology | 2007 | | 1 |
| cpdart0175 | Synthesis and evaluation of 3-phenylpyrazolo[3,4-d]pyrimidine-peptide conjugates as Src kinase inhibitors | Kumar, Anil; Wang, Yuehao; Lin, Xiaofeng; Sun, Gongqin; Parang, Keykavous | ChemMedChem | 2007 | | 13 |
| cpdart0176 | Synthesis of a pyridoxine-peptide based delivery system for nucleotides | Marchand, Arnaud; Marchand, Damien; Busson, Roger; Marliere, Philipe; Herdewijn, Piet | Chemistry & Biodiversity | 2007 | | 7 |
| cpdart0177 | Improved anti-osteoporosis potency and reduced endometrial membrane hyperplasia during hormone replacement therapy with estrogen-RGD peptide conjugates | Xiong, Yu; Zhao, Ming; Wang, Chao; Chang, Heng Wei; Peng, Shiqi | Journal of Medicinal Chemistry | 2007 | | 10 |
| cpdart0178 | (p-Sulfomethyl)phenylalanine as a mimic of O-sulfatyl-tyrosine in synthetic partial sequences of P-Selectin glycoprotein ligand 1 (PSGL-1) | Herzner, Holger; Kunz, Horst | Tetrahedron | 2007 | | 3 |
| cpdart0179 | Synthesis and Binding Studies of Alzheimer Ligands on Solid Support | Rzepecki, Petra; Geib, Nina; Peifer, Manuel; Biesemeier, Frank; Schrader, Thomas | Journal of Organic Chemistry | 2007 | | 9 |
| cpdart0180 | Synthesis of Biologically Active Peptide Nucleic Acid-Peptide Conjugates by Sortase-Mediated Ligation | Pritz, Stephan; Wolf, Yvonne; Kraetke, Oliver; Klose, Jana; Bienert, Michael; Beyermann, Michael | Journal of Organic Chemistry | 2007 | | 20 |
| cpdart0181 | A Peptide Conjugate of Vitamin E Succinate Targets Breast Cancer Cells with High ErbB2 Expression | Wang, Xiu-Fang; Birringer, Marc; Dong, Lan-Feng; Veprek, Pavel; Low, Pauline; Swettenham, Emma; Stantic, Marina; Yuan, Lin-Hong; Zobalova, Renata; Wu, Kun; Ledvina, Miroslav; Ralph, Stephen J.; Neuzil, Jiri | Cancer Research | 2007 | | 1 |
| cpdart0182 | Spacer-separated sialyl Lewisx cyclo-peptide conjugates as potential E-selectin ligands | Herzner, Holger; Kunz, Horst | Carbohydrate Research | 2007 | | 2 |
| cpdart0183 | The use of fullerene substituted phenylalanine amino acid as a passport for peptides through cell membranes | Yang, Jianzhong; Wang, Kuan; Driver, Jonathan; Yang, Jianhua; Barron, Andrew R. | Organic & Biomolecular Chemistry | 2007 | | 5 |
| cpdart0184 | Bifunctional ligands that target cells displaying the αvβ3 integrin | Owen, Robert M.; Carlson, Coby B.; Xu, Jinwang; Mowery, Patricia; Fasella, Elisabetta; Kiessling, Laura L. | ChemBioChem | 2007 | | 4 |
| cpdart0185 | AZT and AZT-monophosphate prodrugs incorporating HIV-protease substrate fragment: synthesis and evaluation as specific drug delivery systems | Liotard, Jean-Francois; Mehiri, Mohamed; Di Giorgio, Audrey; Boggetto, Nicole; Reboud-Ravaux, Michele; Aubertin, Anne-Marie; Condom, Roger; Patino, Nadia | Antiviral Chemistry & Chemotherapy | 2006 | | 28 |
| cpdart0186 | Acridin-9-yl exchange: a proposal for the action of some 9-aminoacridine drugs | Sebestik, Jaroslav; Safarik, Martin; Stibor, Ivan; Hlavacek, Jan | Biopolymers | 2006 | | 2 |
| cpdart0187 | REPLACE: a strategy for iterative design of cyclin-binding groove inhibitors | Andrews, Martin J. I.; Kontopidis, George; McInnes, Campbell; Plater, Andy; Innes, Lorraine; Cowan, Angela; Jewsbury, Philip; Fischer, Peter M. | ChemBioChem | 2006 | | 17 |
| cpdart0188 | Delivery of 2-5A cargo into living cells using the Tat cell penetrating peptide: 2-5A-tat | Zhou, Longhu; Thakur, Chandar S.; Molinaro, Ross J.; Paranjape, Jayashree M.; Hoppes, Rieuwert; Jeang, Kuan-Teh; Silverman, Robert H.; Torrence, Paul F. | Bioorganic & Medicinal Chemistry | 2006 | | 4 |
| cpdart0189 | Improved Therapeutic Efficacy of Doxorubicin through Conjugation with a Novel Peptide Drug Delivery Technology (Vectocell) | Meyer-Losic, Florence; Quinonero, Jerome; Dubois, Vincent; Alluis, Bertrand; Dechambre, Mireille; Michel, Matthieu; Cailler, Francoise; Fernandez, Anne-Marie; Trouet, Andre; Kearsey, Jonathan | Journal of Medicinal Chemistry | 2006 | | 7 |
| cpdart0190 | Dual-acting agents that possess free radical scavenging and antithrombotic activities: Design, synthesis, and evaluation of phenolic tetrahydro-β-carboline RGD peptide conjugates | Bi, Wei; Bi, Lanrong; Cai, Jianhui; Liu, Sanguang; Peng, Shiqi; Fischer, Nicholas O.; Tok, Jeffrey B.-H.; Wang, Guohua | Bioorganic & Medicinal Chemistry | 2006 | | 6 |
| cpdart0191 | Turn and helical peptide spacers: combined distance and angular dependencies in the exciton-coupled circular dichroism of intramolecularly interacting bis-porphyrins | Guryanov, Ivan; Moretto, Alessandro; Campestrini, Sandro; Broxterman, Quirinus B.; Kaptein, Bernard; Peggion, Cristina; Formaggio, Fernando; Toniolo, Claudio | Biopolymers | 2006 | | 13 |
| cpdart0192 | New peptide conjugates with 9-aminoacridine: synthesis and binding to DNA | Sebestik, Jaroslav; Stibor, Ivan; Hlavacek, Jan | Journal of Peptide Science | 2006 | | 7 |
| cpdart0193 | Single-Drug Multiligand Conjugates: Synthesis and Preliminary Cytotoxicity Evaluation of a Paclitaxel-Dipeptide "Scorpion"" Molecule" | Safavy, Ahmad; Raisch, Kevin P.; Matusiak, Damien; Bhatnagar, Saloni; Helson, Lawrence | Bioconjugate Chemistry | 2006 | | 2 |
| cpdart0194 | Phosphorylation State-Responsive Lanthanide Peptide Conjugates: A Luminescence Switch Based on Reversible Complex Reorganization | Tremblay, Matthew S.; Zhu, Qing; Marti, Angel A.; Dyer, Joanne; Halim, Marlin; Jockusch, Steffen; Turro, Nicholas J.; Sames, Dalibor | Organic Letters | 2006 | | 2 |
| cpdart0195 | Synthesis of oligotuftsin-based branched oligopeptide conjugates for chemotactic drug targeting | Mezo, Gabor; Lang, Orsolya; Jakab, Annamaria; Bai, Katalin B.; Szabo, Ildiko; Schlosser, Gitta; Lang, Julianna; Kohidai, Laszlo; Hudecz, Ferenc | Journal of Peptide Science | 2006 | | 3 |
| cpdart0196 | Peptide-doxorubicin conjugates specifically degraded by matrix metalloproteinases expressed from tumor | Lee, Gee Young; Song, Ji-hye; Kim, Sang Yoon; Park, Kyeongsoon; Byun, Youngro | Drug Development Research | 2006 | | 6 |
| cpdart0197 | Synthesis and biological activity of conjugates between paclitaxel and the cell delivery vector penetratin | Wang, Shudong; Zhelev, Nikolai Z.; Duff, Susan; Fischer, Peter M. | Bioorganic & Medicinal Chemistry | 2006 | | 6 |
| cpdart0198 | Design of an IV Formulation of an Unstable Prodrug Candidate for Prostate Cancer Treatment: Solution Chemistry of N-(glutaryl-hyp-ala-ser-cyclohexylglycyl-gln-ser-leu)-doxorubicin | Karki, Shyam; Treemaneekarn, Varaporn; Ostovic, Drazen; Nerurkar, Maneesh; Almarsson, Oern | Drug Development and Industrial Pharmacy | 2006 | | 1 |
| cpdart0199 | Peptide-Mediated Cell Transport of Water Soluble Porphyrin Conjugates | Sibrian-Vazquez, Martha; Jensen, Timothy J.; Hammer, Robert P.; Vicente, M. Graca H. | Journal of Medicinal Chemistry | 2006 | | 5 |
| cpdart0200 | Synthesis of acridine-nuclear localization signal (NLS) conjugates and evaluation of their impact on lipoplex and polyplex-based transfection | Boulanger, Caroline; Di Giorgio, Christophe; Vierling, Pierre | European Journal of Medicinal Chemistry | 2005 | | 4 |
| cpdart0201 | Synthesis and characterization of positively charged porphyrin-peptide conjugates | Sibrian-Vazquez, Martha; Jensen, Timothy J.; Fronczek, Frank R.; Hammer, Robert P.; Vicente, M. Graca H. | Bioconjugate Chemistry | 2005 | | 10 |
| cpdart0202 | Mechanism and structure-activity relationships of norspermidine-based peptidic inhibitors of trypanothione reductase | Dixon, Mark J.; Maurer, Richard I.; Biggi, Cristina; Oyarzabal, Julen; Essex, Jonathan W.; Bradley, Mark | Bioorganic & Medicinal Chemistry | 2005 | | 2 |
| cpdart0203 | Synthesis and Biological Activity of Nitronyl Nitroxide Containing Peptides | Zhao, Ming; Liu, Junling; Wang, Chao; Wang, Lili; Liu, Hu; Peng, Shiqi | Journal of Medicinal Chemistry | 2005 | | 11 |
| cpdart0204 | Self-Assembling Porphyrin-Modified Peptides | Dunetz, Joshua R.; Sandstrom, Claire; Young, Elizabeth R.; Baker, Paul; Van Name, Steven A.; Cathopolous, Terry; Fairman, Robert; De Paula, Julio C.; Kerfeldt, Karin S. | Organic Letters | 2005 | | 1 |
| cpdart0205 | One pot conjugation of the polypeptides directed by phosphorus oxychloride | Zhou, N.; Liu, Y.; Zhou, G. J.; Zhao, Y. F. | Journal of Peptide Research | 2005 | | 18 |
| cpdart0206 | Synthesis, Characterization, and Cellular Uptake of DNA-Binding Rose Bengal Peptidoconjugates | Carreon, Jay R.; Roberts, Marcel A.; Wittenhagen, Lisa M.; Kelley, Shana O. | Organic Letters | 2005 | | 7 |
| cpdart0207 | DNA scission chemistry and EPR studies of four new bis(2,6-dimethoxyhydroquinone-3-mercaptoacetic acid)-peptide conjugates | Song, Yu-Fei | Australian Journal of Chemistry | 2004 | | 4 |
| cpdart0208 | Synthesis of a silk-inspired peptide-oligothiophene conjugate | Klok, Harm-Anton; Roesler, Annette; Goetz, Guenther; Mena-Osteritz, Elena; Baeuerle, Peter | Organic & Biomolecular Chemistry | 2004 | | 1 |
| cpdart0209 | Synthesis and Characterization of Peptide-Cationic Steroid Antibiotic Conjugates | Ding, Bangwei; Taotofa, Uale; Orsak, Thomas; Chadwell, Matthew; Savage, Paul B. | Organic Letters | 2004 | | 9 |
| cpdart0210 | The synthesis and immunosuppressive activities of steroid-urotoxin linkers | Wang, Chao; Zhao, Ming; Qiu, Xuecai; Peng, Shiqi | Bioorganic & Medicinal Chemistry | 2004 | | 13 |
| cpdart0211 | De novo design, synthesis, and function of semiartificial myoglobin conjugated with coiled-coil two-α-helix peptides | Sakamoto, Seiji; Ito, Atsushi; Kudo, Kazuaki; Yoshikawa, Susumu | Chemistry - A European Journal | 2004 | | 3 |
| cpdart0212 | 2-Pyrrolinodoxorubicin and its peptide-vectorized form bypass multidrug resistance | Castex, Cedric; Merida, Peggy; Blanc, Emmanuelle; Clair, Philippe; Rees, Anthony R.; Temsamani, Jamal | Anti-Cancer Drugs | 2004 | | 3 |
| cpdart0213 | Arginine carrier peptide bearing Ni(II) chelator to promote cellular uptake of histidine-tagged proteins | Futaki, Shiroh; Niwa, Miki; Nakase, Ikuhiko; Tadokoro, Akiko; Zhang, Youjun; Nagaoka, Makoto; Wakako, Naoya; Sugiura, Yukio | Bioconjugate Chemistry | 2004 | | 5 |
| cpdart0214 | Efficient synthesis of RGD-containing cyclic peptide-porphyrin conjugates by ring-closing metathesis on solid support | Chaleix, Vincent; Sol, Vincent; Guilloton, Michel; Granet, Robert; Krausz, Pierre | Tetrahedron Letters | 2004 | | 6 |
| cpdart0215 | Design, synthesis, and characterization of an ATP-peptide conjugate inhibitor of protein kinase A | Hines, Aliya C.; Cole, Philip A. | Bioorganic & Medicinal Chemistry Letters | 2004 | | 3 |
| cpdart0216 | Thiazole orange-peptide conjugates: Sensitivity of DNA binding to chemical structure | Carreon, Jay R.; Mahon, Kerry P. Jr.; Kelley, Shana O. | Organic Letters | 2004 | | 4 |
| cpdart0217 | Zipper-Featured δ-Peptide Foldamers Driven by Donor-Acceptor Interaction. Design, Synthesis, and Characterization | Zhao, Xin; Jia, Mu-Xin; Jiang, Xi-Kui; Wu, Li-Zhu; Li, Zhan-Ting; Chen, Guang-Ju | Journal of Organic Chemistry | 2004 | | 9 |
| cpdart0218 | HPLC-MS/MS determination of a peptide conjugate prodrug of doxorubicin, and its active metabolites, leucine-doxorubicin and doxorubicin, in dog and rat plasma | Mazuel, Claude; Grove, Jeffrey; Gerin, Genevieve; Keenan, Kevin P. | Journal of Pharmaceutical and Biomedical Analysis | 2003 | | 2 |
| cpdart0219 | Toward Artificial Developmental Regulators | Arndt, Hans-Dieter; Hauschild, Karl E.; Sullivan, David P.; Lake, Kara; Dervan, Peter B.; Ansari, Aseem Z. | Journal of the American Chemical Society | 2003 | | 2 |
| cpdart0220 | Receptor-Mediated Targeting of a Photosensitizer by Its Conjugation to Gonadotropin-Releasing Hormone Analogues | Rahimipour, Shai; Ben-Aroya, Nurit; Ziv, Keren; Chen, Alon; Fridkin, Mati; Koch, Yitzhak | Journal of Medicinal Chemistry | 2003 | | 2 |
| cpdart0221 | Self-Assembling of the Porphyrin-Linked Acyclic Penta- and Heptapeptides in Aqueous Trifluoroethanol | Arai, Toru; Inudo, Makiko; Ishimatsu, Tomomi; Akamatsu, Chieko; Tokusaki, Yasushi; Sasaki, Tomikazu; Nishino, Norikazu | Journal of Organic Chemistry | 2003 | | 3 |
| cpdart0222 | An efficient synthesis of a doxorubicin-peptide conjugate | Shi, Yao-Jun; Cameron, Mark; Dolling, Ulf H.; Lieberman, David R.; Lynch, Joseph E.; Reamer, Robert A.; Robbins, Michael A.; Volante, R. P.; Reider, Paul J. | Synlett | 2003 | | 1 |
| cpdart0223 | New dsDNA-binding hybrid molecules combining an unnatural peptide and an intercalating moiety | Chaltin, Patrick; Borgions, Filip; Rozenski, Jef; Van Aerschot, Arthur; Herdewijn, Piet | Helvetica Chimica Acta | 2003 | | 23 |
| cpdart0224 | An adjustable release rate linking strategy for cytotoxin-Peptide conjugates | Fuselier, Joseph A.; Sun, Lichun; Woltering, S. Nathaniel; Murphy, William A.; Vasilevich, Natalya; Coy, David H. | Bioorganic & Medicinal Chemistry Letters | 2003 | | 6 |
| cpdart0225 | Amino acid and peptide conjugates of protoporphyrin: preparation and analysis by high-performance liquid chromatography, high-performance liquid chromatography/electrospray ionization mass spectrometry and matrix-assisted laser desorption/ionization time-of-flight mass spectrometry | Razzaque, M. A.; Lord, G. A.; Lim, C. K. | Rapid Communications in Mass Spectrometry | 2002 | | 7 |
| cpdart0226 | DNA Cross-Linking with Metallointercalator-Peptide Conjugates | Copeland, Kimberly D.; Lueras, Alexis M. K.; Stemp, Eric D. A.; Barton, Jacqueline K. | Biochemistry | 2002 | | 12 |
| cpdart0227 | Investigations into the chromatographic behavior of a doxorubicin-peptide conjugate | Hicks, Michael B.; Antonucci, Vincent L.; Riddle, Lance; Novak, Tom J.; Skrdla, Peter | Journal of Chromatography A | 2002 | | 1 |
| cpdart0228 | Design and Synthesis of a Pro-Drug of Vinblastine Targeted at Treatment of Prostate Cancer with Enhanced Efficacy and Reduced Systemic Toxicity | Brady, Stephen F.; Pawluczyk, Joseph M.; Lumma, Patricia K.; Feng, Dong-Mei; Wai, Jenny M.; Jones, Raymond; DeFeo-Jones, Deborah; Wong, Bradley K.; Miller-Stein, Cynthia; Lin, Jiunn H.; Oliff, Allen; Freidinger, Roger M.; Garsky, Victor M. | Journal of Medicinal Chemistry | 2002 | | 5 |
| cpdart0229 | Advanced Synthesis & Catalysis | Mann, Enrique; Chana, Antonio; Sanchez-Sancho, Francisco; Puerta, Carmen; Garcia-Merino, Antonio; Herradon, Bernardo | Advanced Synthesis & Catalysis | 2002 | | 9 |
| cpdart0230 | Solid-Phase Synthesis of Symmetrical 3,6-Bispeptide-Acridone Conjugates | Ladame, Sylvain; Harrison, R. John; Neidle, Stephen; Balasubramanian, Shankar | Organic Letters | 2002 | | 4 |
| cpdart0231 | Employment of on-line FT-IR spectroscopy to monitor the deprotection of a 9-fluorenylmethyl protected carboxylic acid peptide conjugate of doxorubicin | Cameron, Mark; Zhou, George X.; Hicks, Micheal B.; Antonucci, Vincent; Ge, Zhihong; Lieberman, David R.; Lynch, Joesph E.; Shi, Yao-Jun | Journal of Pharmaceutical and Biomedical Analysis | 2002 | | 4 |
| cpdart0232 | Characterization of a novel prostate-specific antigen-activated peptide-doxorubicin conjugate in patients with prostate cancer | DiPaola, Robert S.; Rinehart, John; Nemunaitis, John; Ebbinghaus, Scott; Rubin, Eric; Capanna, Terry; Ciardella, Marie; Doyle-Lindrud, Susan; Goodwin, Susan; Fontaine, Michelle; Adams, Ned; Williams, Adrienne; Schwartz, Michael; Winchell, Greg; Wickersham, Karen; Deutsch, Paul; Yao, Siu-Long | Journal of Clinical Oncology | 2002 | | 1 |
| cpdart0233 | Targeted Type 1 phototherapeutic agents using azido-peptide bioconjugates | Rajagopalan, Raghavan; Achilefu, Samuel I.; Jimenez, Hermo N.; Webb, Elizabeth G.; Schmidt, Michelle A.; Bugaj, Joseph E.; Dorshow, Richard B. | International Society for Optical Engineering | 2001 | | 5 |
| cpdart0234 | Preparative Biochemistry & Biotechnology | Song, Y. F.; Yang, P. | Preparative Biochemistry & Biotechnology | 2001 | | 8 |
| cpdart0235 | The Synthesis of a Prodrug of Doxorubicin Designed to Provide Reduced Systemic Toxicity and Greater Target Efficacy | Garsky, Victor M.; Lumma, Patricia K.; Feng, Dong-Mei; Wai, Jenny; Ramjit, Harri G.; Sardana, Mohinder K.; Oliff, Allen; Jones, Raymond E.; DeFeo-Jones, Deborah; Freidinger, Roger M. | Journal of Medicinal Chemistry | 2001 | | 13 |
| cpdart0236 | Improvement of Porphyrin Cellular Delivery and Activity by Conjugation to a Carrier Peptide | Chaloin, Laurent; Bigey, Pascal; Loup, Christophe; Marin, Mariana; Galeotti, Nathalie; Piechaczyk, Marc; Heitz, Frederic; Meunier, Bernard | Bioconjugate Chemistry | 2001 | | 2 |
| cpdart0237 | Anthraquinone-peptides as inhibitors of AP-1 transcription factor | Ijaz, T.; Tran, P.; Ruparelia, K. C.; Teesdale-Spittle, P. H.; Orr, S.; Patterson, L. H. | Bioorganic & Medicinal Chemistry Letters | 2001 | | 8 |
| cpdart0238 | Determinants for the drug release from T-0128, camptothecin analog-carboxymethyl dextran conjugate | Harada, M.; Sakakibara, H.; Yano, T.; Suzuki, T.; Okuno, S. | Journal of Controlled Release | 2000 | | 9 |
| cpdart0239 | Preparation and biological activity of amino acid and peptide conjugates of antitumor hydroxymethylacylfulvene | McMorris, Trevor C.; Yu, Jian; Ngo, Huan-Tony; Wang, Haixia; Kelner, Michael J. | Journal of Medicinal Chemistry | 2000 | | 4 |
| cpdart0240 | Solid-phase synthesis of acridine-peptide conjugates and their analysis by tandem mass spectrometry | Carlson, Coby B.; Beal, Peter A. | Organic Letters | 2000 | | 3 |
| cpdart0241 | Highly parallel nano-synthesis of cleavable peptide-dye conjugates on cellulose membranes | Licha, Kai; Bhargava, Sarah; Rheinlander, Christiane; Becker, Andreas; Schneider-Mergener, Jens; Volkmer-Engert, Rudolf | Tetrahedron Letters | 2000 | | 2 |
| cpdart0242 | Synthesis of porphyrin α,ω-bis(methylamino)peptide constructs | Matthews, Susan E.; Pouton, Colin W.; Threadgill, Michael D. | New Journal of Chemistry | 1999 | | 9 |
| cpdart0243 | Cancer chemotherapy based on targeting of cytotoxic peptide conjugates to their receptors on tumors | Schally, Andrew V.; Nagy, Attila | European Journal of Endocrinology | 1999 | | 1 |
| cpdart0244 | Synthesis of the palmitoylated and prenylated C-terminal lipopeptides of the human R- and N-Ras proteins | Schmittberger, T.; Waldmann, H. | Bioorganic & Medicinal Chemistry | 1999 | | 20 |
| cpdart0245 | A calixarene with four peptide loops: an antibody mimic for recognition of protein surfaces | Hamuro, Yoshitomo; Calama, Mercedes Crego; Park, Hyung Soon; Hamilton, Andrew D. | Angewandte Chemie, International Edition in English | 1997 | | 4 |
| cpdart0246 | Benzenesulfonamide-peptide conjugates as probes for secondary binding sites near the active site of carbonic anhydrase | Sigal, George B.; Whitesides, George M. | Bioorganic & Medicinal Chemistry Letters | 1996 | | 43 |
| cpdart0247 | Synthesis of carboxymethylpullulan-peptide-doxorubicin conjugates and their properties | Nogusa, Hideo; Yano, Toshiro; Okuno, Satoshi; Hamana, Hiroshi; Inoue, Kazuhiro | Chemical & Pharmaceutical Bulletin | 1995 | | 1 |
| cpdart0248 | Synthesis and immunological evaluation of the conjugates composed of a muramyl peptide GMDP and tuftsin | Titov, Vladimir M.; Meshcheryakova, Elena A.; Balashova, Tamara A.; Andronova, Tatyana M.; Ivanov, Vadim T. | International Journal of Peptide & Protein Research | 1995 | | 4 |
| cpdart0249 | A Bioactive Fullerene Peptide | Toniolo, Claudio; Bianco, Alberto; Maggini, Michele; Scorrano, Gianfranco; Prato, Maurizio; Marastoni, Mauro; Tomatis, Roberto; Spisani, Susanna; Palu, Giorgio; Blair, Edward D. | Journal of Medicinal Chemistry | 1994 | | 1 |
| cpdart0250 | Preparation of Vitamin B6-Conjugated Peptides at the Amino Terminus and of Vitamin B6-Peptide-Oligonucleotide Conjugates | Zhu, Tianmin; Stein, Stanley | Bioconjugate Chemistry | 1994 | | 1 |
| cpdart0251 | Studies of N-terminal templates for α-helix formation. Synthesis and conformational analysis of peptide conjugates of (2S,5S,8S,11S)-1-acetyl-1,4-diaza-3-keto-5-carboxy-10-thiatricyclo[2.8.1.04,8]tridecane (Ac-Hel1-OH) | Kemp, D. S.; Curran, Timothy P.; Boyd, James G.; Allen, Thomas J. | Journal of Organic Chemistry | 1991 | | 10 |
