Synthesis of peptide conjugates of mestranol by a 1,3-dipolar cycloaddition click reaction

Authors: Sokolova, N. V.; Nenajdenko, V. G.; Chemistry of Heterocyclic Compounds; (2012); 10.1007/s10593-012-1074-3

An efficient method is presented for the synthesis of a series of peptide conjugates of the ethynylestradiol 3-methyl ether and the corresponding azidopeptides by a copper(I)-catalyzed 1,3-di-polar cycloaddition click reaction.

Cpdart0107