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View Conjugates details

ConjuPepDB ID: cpd01525

Chemical structure


molecule
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cpd01525


Schematic Help Icon Schematic representation of peptide, linker and drug in the peptide-drug conjugates
MGLGLHLLVLAAALQGAKKKRKV mercaptoacetic acid Porfirin derivative
Identification
ConjuPepDB ID

cpd01525

Smiles
Molecular weight

3343.8

Molecular formula

C163H247MnN42O27S2

Peptide information
Sequence (one letter)

MGLGLHLLVLAAALQGAKKKRKV

Length

23

Peptide name

amphipathic signal-nuclear localization peptide combination

External ID
CAS number

370102-46-8

Other information
Application

Anticancer therapy, DNA cleavage

Additional function

Improve cellular delivery and activity

Pharmacological class

anticancer

Conjugate type

amide

Linker

N/A

Linker Type

mercaptoacetic acid

Small molecule

Porfirin derivative

Small molecule CAS

370100-96-2

Structure method

HPLC

Rotatable bonds

102

Citations
ID Title Year Authors Journal DOI

cpdart0236

Improvement of Porphyrin Cellular Delivery and Activity by Conjugation to a Carrier Peptide

2001

Chaloin, Laurent; Bigey, Pascal; Loup, Christophe; Marin, Mariana; Galeotti, Nathalie; Piechaczyk, Marc; Heitz, Frederic; Meunier, Bernard

Bioconjugate Chemistry

..