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Schematic representation of peptide, linker and drug in the peptide-drug conjugates
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|---|---|---|---|---|
| GGGPKKKXKVGG | triazole | (T-4)-[4-[(3,5-dimethyl-1H-pyrrol-2-yl-κN)(3,5-dimethyl-2H-pyrrol-2-ylidene-κN)methyl]phenolato]difluoro-boron |
| Identification | |
|---|---|
| ConjuPepDB ID | cpd00967 |
| Smiles | |
| Molecular weight | 2507.35 |
| Molecular formula | C121H181BF2N28O25S | Peptide information |
| Sequence (one letter) | GGGPKKKXKVGG |
| Length | 12 |
| Peptide name | N/A |
| External ID | |
|---|---|
| CAS number | 1202406-15-2 |
| Other information | |
|---|---|
| Application | Anticancer therapy |
| Pharmacological class | anticancer |
| Conjugate type | triazole |
| Linker | N/A |
| Linker Type | triazole |
| Small molecule | (T-4)-[4-[(3,5-dimethyl-1H-pyrrol-2-yl-κN)(3,5-dimethyl-2H-pyrrol-2-ylidene-κN)methyl]phenolato]difluoro-boron |
| Small molecule CAS | 870992-10-2 |
71
| Citations | |||||
|---|---|---|---|---|---|
| ID | Title | Year | Authors | Journal | DOI |
Design and synthesis of novel histone deacetylase inhibitor derived from nuclear localization signal peptide | 2009 | Joshua C.Canzoneri; Po C.Chen; Adegboyega K.Oyelere | Bioorganic & Medicinal Chemistry Letters | ||
