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Article ID ▲/▼Title ▲/▼Authors ▲/▼JournalYear ▲/▼ DOI Records
cpdart0001Accumulation of arginine-rich cell-penetrating peptides in tumors and the potential for anticancer drug delivery in vivo.Nakase, Ikuhiko; Konishi, Yusuke; Ueda, Masashi; Saji, Hideo; Futaki, ShirohJournal of controlled release : official journal of the Controlled Release Society2012 1
cpdart0005Design and biological evaluation of cell-penetrating peptide-doxorubicin conjugates as prodrugs.Nasrolahi Shirazi, Amir; Tiwari, Rakesh; Chhikara, Bhupender S; Mandal, Dindyal; Parang, KeykavousMolecular pharmaceutics2013 2
cpdart0012Controlled release of free doxorubicin from peptide-drug conjugates by drug loading.Chen, Zhipeng; Zhang, Pengcheng; Cheetham, Andrew G; Moon, Jae Hyon; Moxley, James W Jr; Lin, Yi-an; Cui, HonggangJournal of controlled release : official journal of the Controlled Release Society2014 3
cpdart0014Cell penetrating peptides as efficient nanocarriers for delivery of antifungal compound, natamycin for the treatment of fungal keratitis.Jain, Aastha; Shah, Sushmita G; Chugh, ArchanaPharmaceutical research2015 1
cpdart0015Activable Cell-Penetrating Peptide Conjugated Prodrug for Tumor Targeted Drug Delivery.Cheng, Hong; Zhu, Jing-Yi; Xu, Xiao-Ding; Qiu, Wen-Xiu; Lei, Qi; Han, Kai; Cheng, Yin-Jia; Zhang, Xian-ZhengACS Applied Materials & Interfaces2015 1
cpdart0016Dual-targeting hybrid peptide-conjugated doxorubicin for drug resistance reversal in breast cancer.Sheng, Yuan; You, Yiwen; Chen, YunInternational Journal of Pharmaceutics2016 1
cpdart0020BH3 mimetics derived from Bim-BH3 domain core region show PTP1B inhibitory activity.Lu, Xiao; Wu, Lijuan; Liu, Xiaochun; Wang, Shulin; Zhang, ChuanliangBioorganic and Medicinal Chemistry Letters2019 1
cpdart0021Increasing the potential of cell-penetrating peptides for cancer therapy using a new pentagonal scaffold.Duarte, Diana; Fraga, Alexandra G.; Pedrosa, Jorge; Martel, Fátima; Vale, NunoEuropean Journal of Pharmacology2019 6
cpdart0023Novel peptide conjugates for tumor-specific chemotherapy.Langer, Michael; Kratz, Felix; Rothen-Rutishauser, Barbara; Wunderli-Allenspach, Heidi; Beck-Sickinger, Annette G.Journal of Medicinal Chemistry2001 2
cpdart0025Peptide-Drug Conjugate Linked via a Disulfide Bond for Kidney Targeted Drug DeliveryGeng, Qian; Sun, Xun; Gong, Tao; Zhang, Zhi-RongBioconjugate Chemistry2012 2
cpdart0026Cancer chemotherapy based on targeting of cytotoxic peptide conjugates to their receptors on tumorsSchally, Andrew V.; Nagy, AttilaEuropean Journal of Endocrinology1999 1
cpdart0027Design, synthesis and biological evaluation of peptide-NSAID conjugates for targeted cancer therapyShokri, Bahareh; Zarghi, Afshin; Shahhoseini, Soraya; Mohammadi, Reza; Kobarfard, FarzadArchiv der Pharmazie2019 8
cpdart0028Synthesis and anti-cancer evaluation of folic acid-peptide- paclitaxel conjugates for addressing drug resistanceDai, Yuxuan; Cai, Xingguang; Bi, Xinzhou; Liu, Chunxia; Yue, Na; Zhu, Ying; Zhou, Jiaqi; Fu, Mian; Huang, Wenlong; Qian, HaiEuropean Journal of Medicinal Chemistry2019 7
cpdart0029Synthesis and biological evaluation of a novel series of curcumin-peptide derivatives as PepT1-mediated transport drugsZhang, Jiyun; Wen, Hongmei; Shen, Fei; Wang, Xinzhi; Shan, Chenxiao; Chai, Chuan; Liu, Jian; Li, WeiBioorganic Chemistry2019 20
cpdart0030N-Methyl-N-phenylvinylsulfonamides for Cysteine-Selective ConjugationHuang, Rong; Li, Zhihong; Sheng, Yao; Yu, Jianghui; Wu, Yue; Zhan, Yuexiong; Chen, Hongli; Jiang, BiaoOrganic Letters2018 12
cpdart0031Chemoselective Peptide Modification via Photocatalytic Tryptophan β-Position ConjugationYu, Younong; Zhang, Li-Kang; Buevich, Alexei V.; Li, Guoqing; Tang, Haiqun; Vachal, Petr; Colletti, Steven L.; Shi, Zhi-CaiJournal of the American Chemical Society2018 20
cpdart0032Effect of low charge and high hydrophobicity on antimicrobial activity of the quinazolinone-peptide conjugatesRakesh, Kadallipura Puttaswamy; Ramesh, Suhas; Shivakumar; Gowda, Dase ChanneRussian Journal of Bioorganic Chemistry2018 20
cpdart0033In vitro biological evaluation of new antimycobacterial salicylanilide-tuftsin conjugatesEuropean Journal of Medicinal ChemistryEuropean Journal of Medicinal Chemistry2017 22
cpdart0034Enhancing the Potency of Nalidixic Acid toward a Bacterial DNA Gyrase with Conjugated PeptidesAhmed, Marya; Kelley, Shana O.ACS Chemical Biology2017 5
cpdart0035Biological characterization of novel nitroimidazole-peptide conjugates in vitro and in vivoBergmann, Ralf; Splith, Katrin; Pietzsch, Jens; Bachmann, Michael; Neundorf, InesJournal of Peptide Science2017 4
cpdart0036Peptide Conjugates of Benzene Carboxylic Acids as Agonists and Antagonists of Amylin AggregationProfit, Adam A.; Vedad, Jayson; Desamero, Ruel Z. B.Bioconjugate Chemistry2017 9
cpdart0037Truncated Autoinducing Peptide Conjugates Selectively Recognize and Kill Staphylococcus aureusTsuchikama, Kyoji; Shimamoto, Yasuhiro; Anami, YasuakiACS Infectious Diseases2017 13
cpdart0038Cyclic peptide conjugate of curcumin and doxorubicin as an anticancer agentDarwish, Shaban; Mozaffari, Saghar; Parang, Keykavous; Tiwari, RakeshTetrahedron Letters2017 2
cpdart0039Designing Hybrid Antibiotic Peptide Conjugates To Cross Bacterial MembranesDeshayes, Stephanie; Xian, Wujing; Schmidt, Nathan W.; Kordbacheh, Shadi; Lieng, Juelline; Wang, Jennifer; Zarmer, Sandra; Germain, Samantha St.; Voyen, Laura; Thulin, Julia; Wong, Gerard C. L.; Kasko, Andrea M.Bioconjugate Chemistry2017 5
cpdart0040Microwave Energy in Ugi Four-Component Reaction (Ugi-4CR): Expedient Synthesis of Steroid-Peptide Conjugates Based on Aminosteroids - An Important Class of Hybrid SystemsBorah, Preetismita; Chowdhury, Pritish; Begum, AshmaCurrent Organic Synthesis2017 5
cpdart0041Cell-penetrating conjugates of pentaglutamylated methotrexate as potential anticancer drugs against resistant tumor cellsSzabo, Ildiko; Orban, Erika; Schlosser, Gitta; Hudecz, Ferenc; Banoczi, ZoltanEuropean Journal of Medicinal Chemistry2016 7
cpdart0042Design, synthesis, and evaluation of Trolox-conjugated amyloid-β C-terminal peptides for therapeutic intervention in an in vitro model of Alzheimer’s diseaseArai, Takuya; Ohno, Akiko; Kazunori, Mori; Kakizawa, Taeko; Kuwata, Hiroshi; Ozawa, Toshihiko; Shibanuma, Motoko; Hara, Shuntaro; Ishida, Seiichi; Kurihara, Masaaki; Miyata, Naoki; Nakagawa, Hidehiko; Fukuhara, KiyoshiBioorganic & Medicinal Chemistry2016 11
cpdart0043Delivering aminopyridine ligands into cancer cells through conjugation to the cell-penetrating peptide BP16Soler, M.; Gonzalez-Bartulos, M.; Figueras, E.; Massaguer, A.; Feliu, L.; Planas, M.; Ribas, X.; Costas, M.Organic & Biomolecular Chemistry2016 10
cpdart0044Dual Targeting of Intracellular Pathogenic Bacteria with a Cleavable Conjugate of Kanamycin and an Antibacterial Cell-Penetrating PeptideBrezden, Anna; Mohamed, Mohamed F.; Nepal, Manish; Harwood, John S.; Kuriakose, Jerrin; Seleem, Mohamed N.; Chmielewski, JeanJournal of the American Chemical Society2016 2
cpdart0045An effective conjugation strategy for designing short peptide-based HIV-1 fusion inhibitorsLiang, Guodong; Wang, Huixin; Chong, Huihui; Cheng, Siqi; Jiang, Xifeng; He, Yuxian; Wang, Chao; Liu, KeliangOrganic & Biomolecular Chemistry2016 5
cpdart0046Peptide-assisted enhancement of inhibitory effects of small molecular inhibitors for kinasesWang, Wei; Hirano, Yoshinori; Uzawa, Takanori; Taiji, Makoto; Ito, YoshihiroBulletin of the Chemical Society of Japan2016 1
cpdart0047Linker dependent chirality of solvent induced self-assembled structures of porphyrin–α-helical peptide conjugatesBiscaglia, Francesca; Frezza, Elisa; Zurlo, Enrico; Gobbo, MarinaOrganic & Biomolecular Chemistry2016 10
cpdart0048Design and synthesis of peptide conjugates of phosphoramide mustard as prodrugs activated by prostate-specific antigenWu, Xinghua; Hu, LongqinBioorganic & Medicinal Chemistry2016 6
cpdart0050Intracellular Generation of a Diterpene-Peptide Conjugate that Inhibits 14-3-3-Mediated InteractionsParvatkar, Prakash; Kato, Nobuo; Uesugi, Motonari; Sato, Shin-ichi; Ohkanda, JunkoJournal of the American Chemical Society2015 3
cpdart0051Synthesis, drug release, and biological evaluation of new anticancer drug-bioconjugates containing somatostatin backbone cyclic analog as a targeting moietyRedko, Boris; Ragozin, Elena; Andreii, Bazylevich; Helena, Tuchinsky; Amnon, Albeck; Talia, Shekhter Zahavi; Mor, Oron-Herman; Genady, Kostenich; Gary, GellermanBiopolymers2015 5
cpdart0052Synthesis of a New Peptide-Coumarin Conjugate: A Potential Agent against CryptococcosisFerreira, Soraya Z.; Carneiro, Hellem C.; Lara, Hugo A.; Alves, Rosemeire B.; Resende, Jarbas M.; Oliveira, Heloisa M.; Silva, Luciana M.; Santos, Daniel A.; Freitas, Rossimiriam P.ACS Medicinal Chemistry Letters2015 1
cpdart0053Synthesis of Tridecaptin-Antibiotic Conjugates with in Vivo Activity against Gram-Negative BacteriaCochrane, Stephen A.; Li, Xuefeng; He, Sisi; Yu, Min; Wu, Min; Vederas, John C.Journal of Medicinal Chemistry2015 6
cpdart0055Aminocatalysis-Mediated on-Resin Ugi Reactions: Application in the Solid-Phase Synthesis of N-Substituted and Tetrazolo Lipopeptides and PeptidosteroidsMorales, Fidel E.; Garay, Hilda E.; Munoz, Daniela F.; Augusto, Yarelys E.; Otero-Gonzalez, Anselmo J.; Reyes Acosta, Osvaldo; Rivera, Daniel G.Organic Letters2015 14
cpdart0056Synthesis and Activity of 6″-Deoxy-6″-thio-α-GalCer and Peptide ConjugatesCompton, Benjamin J.; Tang, Ching-wen; Johnston, Karen A.; Osmond, Taryn L.; Hayman, Colin M.; Larsen, David S.; Hermans, Ian F.; Painter, Gavin F.Organic Letters2015 2
cpdart0057Efficient synthesis of peptide and protein functionalized pyrrole-imidazole polyamides using native chemical ligationJanssen, Brian M. G.; van Ommeren, Sven P. F. I.; Merkx, MaartenInternational Journal of Molecular Sciences2015 2
cpdart0058Tetrapeptide-coumarin conjugate 3D networks based on hydrogen-bonded charge transfer complexes: gel formation and dye releaseGuo, Zongxia; Gong, Ruiying; Jiang, Yi; Wan, XiaoboSoft Matter2015 2
cpdart0059Enhancing Accumulation and Penetration of HPMA Copolymer-Doxorubicin Conjugates in 2D and 3D Prostate Cancer Cells via iRGD Conjugation with an MMP-2 Cleavable SpacerPeng, Zheng-Hong; Kopecek, JindrichJournal of the American Chemical Society2015 1
cpdart0060Synthesis of bisarylethyne-peptide conjugatesStrack, Martin; Langklotz, Sina; Bandow, Julia E.; Metzler-Nolte, Nils; Bauke Albada, H.Organic Chemistry Frontiers2015 2
cpdart0061Solid-phase-based synthesis of ureidopyrimidinone-peptide conjugates for supramolecular biomaterialsde Feijter, Isja; Goor, Olga J. G. M.; Hendrikse, Simone I. S.; Comellas-Aragones, Marta; Soentjens, Serge H. M.; Zaccaria, Sabrina; Fransen, Peter P. K. H.; Peeters, Joris W.; Milroy, Lech-Gustav; Dankers, Patricia Y. W.Synlett2015 31
cpdart0062Synthesis of new betulinic acid-peptide conjugates and in vivo and in silico studies of the influence of peptide moieties on the triterpenoid core activityGovdi, Anastasiya I.; Sokolova, Nadezda V.; Sorokina, Irina V.; Baev, Dmitry S.; Tolstikova, Tatyana G.; Mamatyuk, Victor I.; Fadeev, Dmitry S.; Vasilevsky, Sergey F.; Nenajdenko, Valentine G.MedChemComm2015 7
cpdart0063Solid-phase synthesis of peptide conjugates derived from the antimicrobial cyclic decapeptide BPC194Vila, Silvia; Badosa, Esther; Montesinos, Emilio; Feliu, Lidia; Planas, MartaEuropean Journal of Organic Chemistry2015 15
cpdart0064Synthesis and Preliminary Evaluation of Novel Bone-targeting NSAIDs Prodrugs based on Glutamic Acid OligopeptidesZhao, Yi; He, Dongsheng; Ma, Lifang; Guo, LiLetters in Drug Design & Discovery2015 12
cpdart0065Synthesis and mass spectrometry analysis of quaternary cryptando-peptidic conjugatesBachor, Remigiusz; Kluczyk, Alicja; Stefanowicz, Piotr; Szewczuk, ZbigniewJournal of Peptide Science2015 3
cpdart0066Propargyloxyproline regio- and stereoisomers for Click-conjugation of peptides: Synthesis and application in linear and cyclic peptidesNorthfield, Susan E.; Mountford, Simon J.; Wielens, Jerome; Liu, Mengjie; Zhang, Lei; Herzog, Herbert; Holliday, Nicholas D.; Scanlon, Martin J.; Parker, Michael W.; Chalmers, David K.; Thompson, Philip E.Australian Journal of Chemistry2015 25
cpdart0067Ligation of anti-cancer drugs to self-assembling ultrashort peptides by click chemistry for localized therapyReithofer, Michael R.; Chan, Kiat-Hwa; Lakshmanan, Anupama; Lam, Dang Hoang; Mishra, Archana; Gopalan, Began; Joshi, Mangesh; Wang, Shu; Hauser, Charlotte A. E.Chemical Science2014 4
cpdart0068Targeted Delivery of Ubiquitin-Conjugated BH3 Peptide-Based Mcl-1 Inhibitors into Cancer CellsMuppidi, Avinash; Doi, Kenichiro; Edwardraja, Selvakumar; Pulavarti, Surya V. S. R. K.; Szyperski, Thomas; Wang, Hong-Gang; Lin, QingBioconjugate Chemistry2014 1
cpdart0069Enthalpy-driven nuclease-like activity and mechanism of peptide-chlorambucil conjugatesYang, Robin C. K.; Huang, Jonathan T. B.; Chen, Yu-Ling; Hung, Chia-Chun; Liao, Mokai; Yao, Wen-Chen; Chen, Chiu-Heng; Liou, Chien-Chung; Waring, Michael J.; Sheh, LeungOrganic & Biomolecular Chemistry2014 2
cpdart0070Macrolide-Peptide Conjugates as Probes of the Path of Travel of the Nascent Peptides through the RibosomeWashington, Arren Z.; Benicewicz, Derek B.; Canzoneri, Joshua C.; Fagan, Crystal E.; Mwakwari, Sandra C.; Maehigashi, Tatsuya; Dunham, Christine M.; Oyelere, Adegboyega K.ACS Chemical Biology2014 8
cpdart0071C60 Pyrrolidine Bis-carboxylic Acid Derivative as a Versatile Precursor for Biocompatible FullerenesAroua, Safwan; Schweizer, W. Bernd; Yamakoshi, YokoOrganic Letters2014 3
cpdart0072Chromatography- and Lyophilization-Free Synthesis of a Peptide-Linker ConjugateMagano, Javier; Bock, Brandon; Brennan, John; Farrand, Douglas; Lovdahl, Michael; Maloney, Mark T.; Nadkarni, Durgesh; Oliver, Wendy K.; Pozzo, Mark J.; Teixeira, John J.; Wang, Jian; Rizzo, John; Tumelty, DavidOrganic Process Research & Development2014 1
cpdart0073Shuttle-Cargo Fusion Molecules of Transport Peptides and the hD2/3 Receptor Antagonist Fallypride: A Feasible Approach To Preserve Ligand-Receptor Binding?Wangler, Carmen; Chowdhury, Shafinaz; Hofner, Georg; Djurova, Petia; Purisima, Enrico O.; Bartenstein, Peter; Wangler, Bjorn; Fricker, Gert; Wanner, Klaus T.; Schirrmacher, RalfJournal of Medicinal Chemistry2014 46
cpdart0074Design, synthesis, and evaluation of derivatives of the fat-accumulation inhibitor ternatin: toward ternatin molecular probesKawazoe, Yoshinori; Tanaka, Yoko; Omura, Sachikazu; Uemura, DaisukeTetrahedron Letters2014 16
cpdart0075Bisubstrate UDP-peptide conjugates as human O-GlcNAc transferase inhibitorsBorodkin, Vladimir S.; Schimpl, Marianne; Gundogdu, Mehmet; Rafie, Karim; Dorfmueller, Helge C.; Robinson, David A.; van Aalten, Daan M. F.Biochemical Journal2014 2
cpdart0076Design, Synthesis and Bioevaluation of an EphA2 Receptor-Based Targeted Delivery SystemBarile, Elisa; Wang, Si; Das, Swadesh K.; Noberini, Roberta; Dahl, Russell; Stebbins, John L.; Pasquale, Elena B.; Fisher, Paul B.; Pellecchia, MaurizioChemMedChem2014 4
cpdart0077Synthesis, Spectroscopic, and Photophysical Characterization and Photosensitizing Activity toward Prokaryotic and Eukaryotic Cells of Porphyrin-Magainin and -Buforin ConjugatesDosselli, Ryan; Ruiz-Gonzalez, Ruben; Moret, Francesca; Agnolon, Valentina; Compagnin, Chiara; Mognato, Maddalena; Sella, Valentina; Agut, Montserrat; Nonell, Santi; Gobbo, Marina; Reddi, ElenaJournal of Medicinal Chemistry2014 5
cpdart0078Design, Synthesis, and Biological Evaluation of Highly Potent Small Molecule-Peptide Conjugates as New HIV-1 Fusion InhibitorsWang, Chao; Shi, Weiguo; Cai, Lifeng; Lu, Lu; Wang, Qian; Zhang, Tianhong; Li, Jinglai; Zhang, Zhenqing; Wang, Kun; Xu, Liang; Jiang, Xifeng; Jiang, Shibo; Liu, KeliangJournal of Medicinal Chemistry2013 4
cpdart0079Synthesis, enzymatic stability and in vitro cytostatic effect of Daunorubicin-GnRH-III derivative dimersSchreier, Verena Natalie; Mezo, Gabor; Orban, Erika; Duerr, Claudia; Marquardt, Andreas; Manea, MarilenaBioorganic & Medicinal Chemistry Letters2013 6
cpdart0080Thiazolidinone-Peptide Hybrids as Dengue Virus Protease Inhibitors with Antiviral Activity in Cell CultureNitsche, Christoph; Schreier, Verena N.; Behnam, Mira A. M.; Kumar, Anil; Bartenschlager, Ralf; Klein, Christian D.Journal of Medicinal Chemistry2013 60
cpdart0081Phthalocyanine-Peptide Conjugates: Receptor-Targeting Bifunctional Agents for Imaging and Photodynamic TherapyRanyuk, Elena; Cauchon, Nicole; Klarskov, Klaus; Guerin, Brigitte; van Lier, Johan E.Journal of Medicinal Chemistry2013 5
cpdart0082Cellular uptake and cytotoxicity of drug-peptide conjugates regulated by conjugation siteZhang, Pengcheng; Cheetham, Andrew G.; Lock, Lye Lin; Cui, HonggangBioconjugate Chemistry2013 6
cpdart0083Synthesis and Antimalarial Bioassay of Quinine - Peptide ConjugatesPanda, Siva S.; Ibrahim, Mohamed A.; Kuecuekbay, Hasan; Meyers, Marvin J.; Sverdrup, Francis M.; El-Feky, Said A.; Katritzky, Alan R.Chemical Biology & Drug Design2013 4
cpdart0084Cholesterol-peptide hybrids to form liposome-like vesicles for gene deliveryTang, Qiong; Cao, Bin; Wu, Haiyan; Cheng, GangPLoS One2013 4
cpdart0085Cell-Penetrating Bisubstrate-Based Protein Kinase C Inhibitorsvan Wandelen, Loek T. M.; van Ameijde, Jeroen; Ismail-Ali, Ahmed F.; van Ufford, H. C. Quarles; Vijftigschild, Lodewijk A. W.; Beekman, Jeffrey M.; Martin, Nathaniel I.; Ruijtenbeek, Rob; Liskamp, Rob M. J.ACS Chemical Biology2013 3
cpdart0086Betulonic acid-peptide conjugates: synthesis and evaluation of anti-inflammatory activityGovdi, Anastasiya I.; Vasilevsky, Sergei F.; Sokolova, Nadezhda V.; Sorokina, Irina V.; Tolstikova, Tatyana G.; Nenajdenko, Valentine G.Mendeleev Communications2013 6
cpdart0087Peptide conjugates of 4-aminocyclophosphamide as prodrugs of phosphoramide mustard for selective activation by prostate-specific antigen (PSA)Jiang, Yongying; Hu, LongqinBioorganic & Medicinal Chemistry2013 8
cpdart0088Novel water-soluble prodrugs of acyclovir cleavable by the dipeptidyl-peptidase IV (DPP IV/CD26) enzymeDiez-Torrubia, Alberto; Cabrera, Silvia; de Castro, Sonia; Garcia-Aparicio, Carlos; Mulder, Gwenn; De Meester, Ingrid; Camarasa, Maria-Jose; Balzarini, Jan; Velazquez, SonsolesEuropean Journal of Medicinal Chemistry2013 8
cpdart0089Organogels of triterpenoid-tripeptide conjugates: Encapsulation of dye molecules and basicity increase associated with aggregationLu, Jinrong; Gao, Yuxia; Wu, Jindan; Ju, YongRSC Advances2013 2
cpdart0090Peptide-Drug Conjugate Linked via a Disulfide Bond for Kidney Targeted Drug DeliveryGeng, Qian; Sun, Xun; Gong, Tao; Zhang, Zhi-RongBioconjugate Chemistry2012 2
cpdart0091The First Generation of β‐Galactosidase‐Responsive Prodrugs Designed for the Selective Treatment of Solid Tumors in Prodrug MonotherapyLegigan, Thibaut; Clarhaut, Jonathan; Tranoy-Opalinski, Isabelle; Monvoisin, Arnaud; Renoux, Brigitte; Thomas, Mikael; Le Pape, Alain; Lerondel, Stephanie; Papot, SebastienAngewandte Chemie, International Edition2012 2
cpdart0092Cell-penetrating γ-peptide/antimicrobial undecapeptide conjugates with anticancer activityRoses, Cristina; Carbajo, Daniel; Sanclimens, Gloria; Farrera-Sinfreu, Josep; Blancafort, Adriana; Oliveras, Gloria; Cirac, Anna D.; Bardaji, Eduard; Puig, Teresa; Planas, Marta; Feliu, Lidia; Albericio, Fernando; Royo, MiriamTetrahedron2012 2
cpdart0093Modular synthesis of supramolecular ureidopyrimidinone-peptide conjugates using an oxime ligation strategyKieltyka, Roxanne E.; Bastings, Maartje M. C.; van Almen, Geert C.; Besenius, Pol; Kemps, Erwin W. L.; Dankers, Patricia Y. W.Chemical Communications2012 7
cpdart0094Optimization of BACE1 inhibition of tripartite structures by modification of membrane anchors, spacers and pharmacophores - development of potential agents for the treatment of Alzheimer's diseaseLinning, Philipp; Haussmann, Ute; Beyer, Isaak; Weidlich, Sebastian; Schieb, Heinke; Wiltfang, Jens; Klafki, Hans-Wolfgang; Knoelker, Hans-JoachimOrganic & Biomolecular Chemistry2012 17
cpdart0095A general route to xyloglucan-peptide conjugates for the activation of cellulose surfacesAraujo, Ana Catarina; Nakhai, Azadeh; Ruda, Marcus; Slaettegard, Rikard; Gatenholm, Paul; Brumer, HarryCarbohydrate Research2012 3
cpdart0096Synthesis of [12]aneN3-dipeptide conjugates as metal-free DNA nucleasesLi, Zhi-Fen; Chen, Hua-Long; Zhang, Li-Jun; Lu, Zhong-LinBioorganic & Medicinal Chemistry Letters2012 8
cpdart0097DOTA-tris(OPp ester) as a bifunctional prochelator for the preparation of DOTA-peptide conjugatesJamous, Mazen; Haberkorn, Uwe; Mier, WalterTetrahedron Letters2012 3
cpdart0098Efficient formation of heterodimers from peptides and proteins using unsymmetrical polyfluorophenyl esters of dicarboxylic acidsSlosarczyk, Adam T.; Baltzer, LarsJournal of Peptide Science2012 8
cpdart0099Synthesis of small molecule-peptide conjugates as potential whitening agentsLee, Hye-Suk; Shin, Kyong-Hoon; Ryu, Geun-Seok; Chi, Gyeong-Yup; Cho, In-Shik; Kim, Han-YoungBulletin of the Korean Chemical Society2012 18
cpdart0100Enhancing cellular uptake of activable cell-penetrating peptide-doxorubicin conjugate by enzymatic cleavageShi, Nian-Qiu; Gao, Wei; Xiang, Bai; Qi, Xian-RongInternational Journal of Nanomedicine2012 1
cpdart0101β-Lactam-host defence peptide conjugates as antibioticprodrug candidates targeting resistant bacteriaDesgranges, Stephane; Ruddle, Carol C.; Burke, Liam P.; McFadden, Tara M.; O'Brien, John E.; Fitzgerald-Hughes, Deirdre; Humphreys, Hilary; Smyth, Timothy P.; Devocelle, MarcRSC Advances2012 3
cpdart0102Enhanced Cellular Uptake of a New, in Silico Identified Antitubercular Candidate by Peptide ConjugationHorvati, Kata; Bacsa, Bernadett; Szabo, Nora; David, Sandor; Mezo, Gabor; Grolmusz, Vince; Vertessy, Beata; Hudecz, Ferenc; Bosze, SzilviaBioconjugate Chemistry2012 2
cpdart0103Methotrexate-cIBR conjugate for targeting methotrexate to leukocytes: Conjugate stability and in vivo efficacy in suppressing rheumatoid arthritisMajumdar, Sumit; Anderson, Meagan E.; Xu, Christine R.; Yakovleva, Tatyana V.; Gu, Leo C.; Malefyt, Thomas R.; Siahaan, Teruna J.Journal of Pharmaceutical Sciences2012 7
cpdart0104A New Family of Highly Potent Inhibitors of Microbes: Synthesis and Conjugation of Elastin Based Peptides to Piperazine DerivativeSuhas, R.; Chandrashekar, S.; Gowda, D. ChanneInternational Journal of Peptide Research and Therapeutics2012 14
cpdart0105Lipopolysaccharide Neutralizing Peptide-Porphyrin Conjugates for Effective Photoinactivation and Intracellular Imaging of Gram-Negative Bacteria StrainsLiu, Fang; Soh Yan Ni, Annie; Lim, Yingjie; Mohanram, Harini; Bhattacharjya, S.; Xing, BengangBioconjugate Chemistry2012 1
cpdart0106Microwave-assisted formation of peptide-vitamin conjugatesEl-Nachef, Claudia; Bajaj, Kiran; Koblick, Jacqueline; Katritzky, Alan R.European Journal of Organic Chemistry2012 11
cpdart0107Synthesis of peptide conjugates of mestranol by a 1,3-dipolar cycloaddition click reactionSokolova, N. V.; Nenajdenko, V. G.Chemistry of Heterocyclic Compounds2012 6
cpdart0108Synthesis of α-Trifluoromethyl-α-hydroxy Acid-Peptide Conjugates via Click ChemistrySokolova, Nadezhda V.; Vorobyeva, Daria V.; Osipov, Sergey N.; Vasilyeva, Tamara P.; Nenajdenko, Valentine G.Synthesis2012 14
cpdart0109Syntheses of chiral N-(protected) tri- and tetrapeptide conjugatesBajaj, Kiran; Panda, Siva S.; El-Nachef, Claudia; Katritzky, Alan R.Chemical Biology & Drug Design2012 7
cpdart0110Novel cinnamic acid/4-aminoquinoline conjugates bearing non-proteinogenic amino acids: Towards the development of potential dual action antimalarialsPerez, Bianca C.; Teixeira, Catia; Figueiras, Marta; Gut, Jiri; Rosenthal, Philip J.; Gomes, Jose R. B.; Gomes, PaulaEuropean Journal of Medicinal Chemistry2012 17
cpdart0112Biological Evaluation of a Novel Doxorubicin-Peptide Conjugate for Targeted Delivery to EGF Receptor-Overexpressing Tumor CellsAi, Shibin; Duan, Jianli; Liu, Xin; Bock, Stephanie; Tian, Yuan; Huang, ZeboMolecular Pharmaceutics2011 2
cpdart0113A New Daunomycin-Peptide Conjugate: Synthesis, Characterization and the Effect on the Protein Expression Profile of HL-60 Cells in VitroOrban, Erika; Manea, Marilena; Marquadt, Andreas; Banoczi, Zoltan; Csik, Gabriella; Fellinger, Erzsebet; Bosze, Szilvia; Hudecz, FerencBioconjugate Chemistry2011 1
cpdart0114Synthesis of elastin based peptides conjugated to benzisoxazole as a new class of potent antimicrobials - A novel approach to enhance biocompatibilitySuhas, R.; Chandrashekar, S.; Gowda, D. ChanneEuropean Journal of Medicinal Chemistry2011 14
cpdart0115New pemetrexed-peptide conjugates: synthesis, characterization and in vitro cytostatic effect on non-small cell lung carcinoma (NCI-H358) and human leukemia (HL-60) cellsMiklan, Zsanett; Orban, Erika; Banoczi, Zoltan; Hudecz, FerencJournal of Peptide Science2011 6
cpdart0116Synthesis and antibacterial activity of amphiphilic lysine-ligated neomycin B conjugatesBera, Smritilekha; Zhanel, George G.; Schweizer, FrankCarbohydrate Research2011 1
cpdart0117Synthesis and Self-Assembly of Oligo(p-phenylenevinylene) Peptide Conjugates in WaterMba, Miriam; Moretto, Alessandro; Armelao, Lidia; Crisma, Marco; Toniolo, Claudio; Maggini, MicheleChemistry - A European Journal2011 2
cpdart0118Novel β-carboline-tripeptide conjugates attenuate mesenteric ischemia/reperfusion injury in the ratBi, Wei; Bi, Yue; Xue, Ping; Zhang, Yanrong; Gao, Xiang; Wang, Zhibo; Li, Meng; Baudy-Floc'h, Michele; Ngerebara, Nathaniel; Li, Xiaoxu; Gibson, K. Michael; Bi, LanrongEuropean Journal of Medicinal Chemistry2011 36
cpdart0119A new class of β-carboline alkaloid-peptide conjugates with therapeutic efficacy in acute limb ischemia/reperfusion injuryBi, Wei; Bi, Yue; Xue, Ping; Zhang, Yanrong; Gao, Xiang; Wang, Zhibo; Li, Meng; Baudy-Floc'h, Michele; Ngerebara, Nathaniel; Michael Gibson, K.; Bi, LanrongEuropean Journal of Medicinal Chemistry2011 26
cpdart0120Syntheses and DNA binding of new cationic porphyrin-tetrapeptide conjugatesMezo, Gabor; Herenyi, Levente; Habdas, Jan; Majer, Zsuzsa; Mysliwa-Kurdziel, Beata; Toth, Katalin; Csik, GabriellaBiophysical Chemistry2011 2
cpdart0121Solid phase synthesis and biological activity of tuftsin conjugatesKukowska-Kaszuba, Magdalena; Dzierzbicka, Krystyna; Serocki, Marcin; Skladanowski, AndrzejJournal of Medicinal Chemistry2011 34
cpdart0123Synthesis and optimization of hyaluronic acid-methotrexate conjugates to maximize benefit in the treatment of osteoarthritisHomma, Akie; Sato, Haruhiko; Tamura, Tatsuya; Okamachi, Akira; Emura, Takashi; Ishizawa, Takenori; Kato, Tatsuya; Matsuura, Tetsu; Sato, Shigeo; Higuchi, Yoshinobu; Watanabe, Tomoyuki; Kitamura, Hidetomo; Asanuma, Kentaro; Yamazaki, Tadao; Ikemi, Masahisa; Kitagawa, Hironoshin; Morikawa, Tadashi; Ikeya, Hitoshi; Maeda, Kazuaki; Takahashi, Koichi; Nohmi, Kenji; Izutani, Noriyuki; Kanda, Makoto; Suzuki, RyohchiBioorganic & Medicinal Chemistry2010 27
cpdart0124Synthesis and in Vitro Antitumor Effect of Vinblastine Derivative-Oligoarginine ConjugatesBanoczi, Zoltan; Gorka-Kereskenyi, Almos; Remenyi, Judit; Orban, Erika; Hazai, Laszlo; Tokesi, Natalia; Olah, Judit; Ovadi, Judit; Beni, Zoltan; Hada, Viktor; Szantay, Csaba Jr.; Hudecz, Ferenc; Kalaus, Gyorgy; Szantay, CsabaBioconjugate Chemistry2010 6
cpdart0125Application of the Dipeptidyl Peptidase IV (DPPIV/CD26) Based Prodrug Approach to Different Amine-Containing DrugsDiez-Torrubia, Alberto; Garcia-Aparicio, Carlos; Cabrera, Silvia; De Meester, Ingrid; Balzarini, Jan; Camarasa, Maria-Jose; Velazquez, SonsolesJournal of Medicinal Chemistry2010 16
cpdart0126Evaluation of amphiphilic aminoglycoside-peptide triazole conjugates as antibacterial agentsBera, Smritilekha; Zhanel, George G.; Schweizer, FrankBioorganic & Medicinal Chemistry2010 13
cpdart0127Synthesis of DOTA-Conjugated Multimeric [Tyr3]Octreotide Peptides via a Combination of Cu(I)-Catalyzed "Click"" Cycloaddition and Thio Acid/Sulfonyl Azide ""Sulfo-Click"" Amidation and Their in Vivo Evaluation"Yim, Cheng-Bin; Dijkgraaf, Ingrid; Merkx, Remco; Versluis, Cees; Eek, Annemarie; Mulder, Gwenn E.; Rijkers, Dirk T. S.; Boerman, Otto C.; Liskamp, Rob M. J.Journal of Medicinal Chemistry2010 4
cpdart0128Synthesis of Mono-ADP-Ribosylated Oligopeptides Using Ribosylated Amino Acid Building Blocksvan der Heden van Noort, Gerbrand J.; van der Horst, Maarten G.; Overkleeft, Herman S.; van der Marel, Gijsbert A.; Filippov, Dmitri V.Journal of the American Chemical Society2010 5
cpdart0129Structural Design, Solid‐Phase Synthesis and Activity of Membrane‐Anchored β‐Secretase Inhibitors on Aβ Generation from Wild‐Type and Swedish‐Mutant APPSchieb, Heinke; Weidlich, Sebastian; Schlechtingen, Georg; Linning, Philipp; Jennings, Gary; Gruner, Margit; Wiltfang, Jens; Klafki, Hans-Wolfgang; Knoelker, Hans-JoachimChemistry - A European Journal2010 9
cpdart0131Biological evaluation of paclitaxel-peptide conjugates as a model for MMP2-targeted drug deliveryYamada, Roppei; Kostova, Maya B.; Anchoori, Ravi Kumar; Xu, Shili; Neamati, Nouri; Khan, Saeed R.Cancer Biology & Therapy2010 3
cpdart0132"Click" synthesis of small molecule-peptide conjugates for organelle-specific delivery and inhibition of lysosomal cysteine proteases"Loh, Yuhui; Shi, Haibin; Hu, Mingyu; Yao, Shao Q.Chemical Communications2010 3
cpdart0133A DOTA-peptide conjugate by copper-free click chemistryMartin, Molly E.; Parameswarappa, Sharavathi G.; O'Dorisio, M. Sue; Pigge, F. Christopher; Schultz, Michael K.Bioorganic & Medicinal Chemistry2010 2
cpdart0134Facile synthesis of peptide-porphyrin conjugates: Towards artificial catalaseUmezawa, Naoki; Matsumoto, Nobuyoshi; Iwama, Shinsuke; Kato, Nobuki; Higuchi, TsunehikoBioorganic & Medicinal Chemistry2010 1
cpdart0135Influence of the number and distribution of NLS peptides on the photosensitizing activity of multimeric porphyrin-NLSSibrian-Vazquez, Martha; Jensen, Timothy J.; Vicente, M. Graca H.Organic & Biomolecular Chemistry2010 3
cpdart0136A Metal-Free DNA Nuclease Based on a Cyclic Peptide ScaffoldAlkhader, Shadad; Ezra, Aviva; Kasparkova, Jana; Brabec, Viktor; Yavin, EylonBioconjugate Chemistry2010 18
cpdart0137Synthesis and Characterization of New Galanthamine Derivatives Comprising Peptide MoietyLyubomir T. Vezenkov, Maria G. Georgieva, Dantcho L. Danalev, Tchavdar B. Ivanov, Galya I. IvanovaProtein & Peptide Letters2009 7
cpdart0138Novel type 1 photosensitizers: viability of leukemia cells exposed to reactive intermediates generated in situ by in vitro photofragmentationRaghavan Rajagopalan, Amol Karwa, Przemyslaw M. Lusiak, Kripa Srivastava, Amruta R. Poreddy, Raghootama S. Pandurangi, Karen P. Galen, William L. Neumann, Gary E. Cantrell, Richard B. DorshowProc. SPIE 7380, Photodynamic Therapy: Back to the Future2009 1
cpdart0139New daunomycin–oligoarginine conjugates: Synthesis, characterization, and effect on human leukemia and human hepatoma cellsZsanett Miklán; Erika Orbán; Gabriella Csík; Gitta Schlosser; Anna Magyar; Ferenc HudeczPeptide Science2009 6
cpdart0140Design and synthesis of novel histone deacetylase inhibitor derived from nuclear localization signal peptideJoshua C.Canzoneri; Po C.Chen; Adegboyega K.OyelereBioorganic & Medicinal Chemistry Letters2009 6
cpdart0141A novel L-ascorbic acid and peptide conjugate with increased stability and collagen biosynthesisHo-Il Choi, Jong-Il Park, Heung-Jae Kim, Dong-Won Kim, Soung-Soo KimBMB Reports2009 1
cpdart0142Peptide Targeting of Platinum Anti-Cancer DrugsNdinguri, Margaret W.; Solipuram, Rajasree; Gambrell, Robert P.; Aggarwal, Sita; Hammer, Robert P.Bioconjugate Chemistry2009 2
cpdart0143Towards the conformational mimicry of the measles virus HNE loop: design, synthesis and biological evaluation of a cyclic bile acid-peptide conjugateBode, Catherine A.; Bechet, Tom; Prodhomme, Emmanuel; Gheysen, Katelijne; Gregoir, Pieter; Martins, Jose C.; Muller, Claude P.; Madder, AnnemiekeOrganic & Biomolecular Chemistry2009 8
cpdart0144An efficient route to VEGF-like peptide porphyrin conjugates via microwave-assisted 'click-chemistry'Bakleh, M. E.; Sol, V.; Estieu-Gionnet, K.; Granet, R.; Deleris, G.; Krausz, P.Tetrahedron2009 2
cpdart0145Synthesis and preliminary evaluation in vitro of novel naproxen-dendritic peptide conjugatesOuyang, Liang; Zhang, Jing; Pan, Junzhu; Yan, Linna; Guo, LiDrug Delivery2009 7
cpdart0146An improved synthesis of releasable luciferin-CPP conjugatesEiriksdottir, Emelia; Langel, Uelo; Rosenthal-Aizman, KatriTetrahedron Letters2009 3
cpdart0147Silver-Catalyzed azaGly Ligation. Application to the Synthesis of Azapeptides and of Lipid-Peptide ConjugatesOllivier, Nathalie; Besret, Soizic; Blanpain, Annick; Melnyk, OlegBioconjugate Chemistry2009 3
cpdart0148Novel hyaluronic acid-methotrexate conjugates for osteoarthritis treatmentHomma, Akie; Sato, Haruhiko; Okamachi, Akira; Emura, Takashi; Ishizawa, Takenori; Kato, Tatsuya; Matsuura, Tetsu; Sato, Shigeo; Tamura, Tatsuya; Higuchi, Yoshinobu; Watanabe, Tomoyuki; Kitamura, Hidetomo; Asanuma, Kentaro; Yamazaki, Tadao; Ikemi, Masahisa; Kitagawa, Hironoshin; Morikawa, Tadashi; Ikeya, Hitoshi; Maeda, Kazuaki; Takahashi, Koichi; Nohmi, Kenji; Izutani, Noriyuki; Kanda, Makoto; Suzuki, RyochiBioorganic & Medicinal Chemistry2009 4
cpdart0149Estrano[17,16-e]pyrimidine-amino acid and estrano[17,16-e]pyrimidine-peptide conjugatesMatsumoto, Tomohiro; Shiine, Kodai; Mataka, Shuntaro; Thiemann, ThiesJournal of Chemical Research2009 7
cpdart0150A new water soluble 3,6,9-trioxaundecanedioic acid-based linker and biotinylating reagentBartos, Adam; Hudecz, Ferenc; Uray, KatalinTetrahedron Letters2009 3
cpdart0151Dipole effects on molecular and electronic structures in a novel conjugate of oligo(phenyleneethynylene) and helical peptideNakayama, Hidenori; Morita, Tomoyuki; Kimura, ShunsakuPhysical Chemistry Chemical Physics2009 2
cpdart01523D QSAR of novel estrogen-RGD peptide conjugates: Getting insight into structural dependence of anti-osteoporosis activity and side effect of estrogen in ERTZhao, Ming; Liu, Jiangyuan; Zhang, Xiaoyi; Peng, Li; Li, Chunyu; Peng, ShiqiBioorganic & Medicinal Chemistry2009 17
cpdart0153Synthesis and stereochemical preference of peptide 4-aminocyclophosphamide conjugates as potential prodrugs of phosphoramide mustard for activation by prostate-specific antigen (PSA)Jiang, Yongying; Di Paola, Robert S.; Hu, LongqinBioorganic & Medicinal Chemistry2009 4
cpdart0154Synthesis, evaluation and 3D QSAR analysis of novel estradiol-RGD octapeptide conjugates with oral anti-osteoporosis activityLiu, Jiangyuan; Zhang, Xiaoyi; Zhao, Ming; Peng, ShiqiEuropean Journal of Medicinal2009 16
cpdart0155Effect of Modification of the Physicochemical Properties of ICAM-1-Derived Peptides on Internalization and Intracellular Distribution in the Human Leukemic Cell Line HL-60Majumdar, Sumit; Tejo, Bimo A.; Badawi, Ahmed H.; Moore, David; Krise, Jeffrey P.; Siahaan, Teruna J.Molecular Pharmaceutics2009 2
cpdart0156Design and efficient synthesis of novel ascorbyl conjugated peptide with high collagen biosynthesis stimulating effectsChoi, Ho-Il; Kim, Heung-Jae; Park, Jong-Il; Shin, Eun-Ho; Kim, Dong-Won; Kim, Soung-SooBioorganic & Medicinal Chemistry Letters2009 2
cpdart0157Synthesis and anti-cancer activity of covalent conjugates of artemisinin and a transferrin-receptor targeting peptideOh, Steve; Kim, Byung Ju; Singh, Narendra P.; Lai, Henry; Sasaki, TomikazuCancer Letters2009 2
cpdart0158Synthesis and Biological Evaluation of Vinca Alkaloids and Phomopsin HybridsNgo, Quoc Anh; Roussi, Fanny; Cormier, Anthony; Thoret, Sylviane; Knossow, Marcel; Guenard, Daniel; Gueritte, FrancoiseJournal of Medicinal Chemistry2009 5
cpdart0159Triple Hybrids of Steroids, Spiroketals, and Oligopeptides as New Biomolecular ChimerasBanerjee, Abhisek; Sergienko, Eduard; Vasile, Stefan; Gupta, Vineet; Vuori, Kristiina; Wipf, PeterOrganic Letters2009 10
cpdart0160Synthesis of daunomycin-oligoarginine conjugates and their effect on human leukemia cells (HL-60)Banoczi, Zoltan; Peregi, Balazs; Orban, Erika; Szabo, Rita; Hudecz, FerencARKIVOC2008 3
cpdart0161Oligo(p-phenylenevinylene)-Peptide Conjugates: Synthesis and Self-Assembly in Solution and at the Solid-Liquid InterfaceMatmour, Rachid; De Cat, Inge; George, Subi J.; Adriaens, Wencke; Leclere, Philippe; Bomans, Paul H. H.; Sommerdijk, Nico A. J. M.; Gielen, Jeroen C.; Christianen, Peter C. M.; Heldens, Jeroen T.; van Hest, Jan C. M.; Loewik, Dennis W. P. M.; De Feyter, Steven; Meijer, E. W.; Schenning, Albertus P. H. J.Journal of the American Chemical Society2008 1
cpdart0162Photoinduced Cytotoxicity and Biodistribution of Prostate Cancer Cell-Targeted PorphyrinsSehgal, Inder; Sibrian-Vazquez, Martha; Vicente, M. Graca H.Journal of Medicinal Chemistry2008 2
cpdart0163In vitro and in vivo evaluation of doxorubicin conjugates with the divalent peptide E-[c(RGDfK)2] that targets integrin αvβ3Ryppa, Claudia; Mann-Steinberg, Hagit; Fichtner, Iduna; Weber, Holger; Satchi-Fainaro, Ronit; Biniossek, Martin L.; Kratz, FelixBioconjugate Chemistry2008 1
cpdart0164A cell-penetrating peptidic GRP78 ligand for tumor cell-specific prodrug therapyYoneda, Yoshiyuki; Steiniger, Sebastian C. J.; Capkova, Katerina; Mee, Jenny M.; Liu, Ying; Kaufmann, Gunnar F.; Janda, Kim D.Bioorganic & Medicinal Chemistry Letters2008 2
cpdart01651-Ethoxyethylidene, a New Group for the Stepwise SPPS of Aminooxyacetic Acid Containing PeptidesFoillard, Stephanie; Ohsten Rasmussen, Martin; Razkin, Jesus; Boturyn, Didier; Dumy, PascalJournal of Organic Chemistry2008 3
cpdart0166Syntheses and cellular studies of water soluble porphyrin-peptide conjugatesSibrian-Vazquez, Martha; Jensen, Timothy J.; Hammer, Robert P.; Vicente, M. Graca H.Proceedings of SPIE-The International Society for Optical Engineering2008 6
cpdart0167Synthesis of a coumarin-histone conjugate for HAT fluorescent assayChen, Ziyue; Zheng, Yujun GeorgeHeterocyclic Communications2008 1
cpdart0168Reversible switching of substrate activity of poly-N-isopropylacrylamide peptide conjugatesMolawi, Kian; Studer, ArmidoChemical Communications2007 7
cpdart0169Efficient conversion of tetrapeptide-based TSAO prodrugs to the parent drug by dipeptidyl-peptidase IV (DPPIV/CD26)Garcia-Aparicio, Carlos; Diez-Torrubia, Alberto; Balzarini, Jan; Lambeir, Anne-Marie; Velazquez, Sonsoles; Camarasa, Maria-JoseAntiviral Research2007 8
cpdart0170Design and synthesis of paclitaxel conjugated with an ErbB2-recognizing peptide, EC-1Li, Peng; Jiang, Sheng; Pero, Stephanie C.; Oligino, Lyn; Krag, David N.; Michejda, Christopher J.; Roller, Peter P.Biopolymers2007 2
cpdart0171Validation of a solid-phase-bound steroid scaffold for the synthesis of novel cyclic peptidosteroidsBode, Catherine A.; Muller, Claude P.; Madder, AnnemiekeJournal of Peptide Science2007 6
cpdart0172Biosynthetic Tailoring of Microcin E492m: Post-translational Modification Affords an Antibacterial Siderophore-Peptide ConjugateNolan, Elizabeth M.; Fischbach, Michael A.; Koglin, Alexander; Walsh, Christopher T.Journal of the American Chemical Society2007 3
cpdart0173Synthesis and antitumor activity of peptide-paclitaxel conjugatesPapas, Serafim; Akoumianaki, Tonia; Kalogiros, Christos; Hadjiarapoglou, Lazaros; Theodoropoulos, Panayiotis A.; Tsikaris, VassiliosJournal of Peptide Science2007 3
cpdart0174Synthesis and assessment of a novel peptide conjugate to deliver phenytoin for wound repairKennedy, C. A.; Chan, F. C.; DeVocelle, M.; Meaney, C.; Bouchier-Hayes, D. J.; Kelly, J. G.Journal of Drug Delivery Science and Technology2007 1
cpdart0175Synthesis and evaluation of 3-phenylpyrazolo[3,4-d]pyrimidine-peptide conjugates as Src kinase inhibitorsKumar, Anil; Wang, Yuehao; Lin, Xiaofeng; Sun, Gongqin; Parang, KeykavousChemMedChem2007 13
cpdart0176Synthesis of a pyridoxine-peptide based delivery system for nucleotidesMarchand, Arnaud; Marchand, Damien; Busson, Roger; Marliere, Philipe; Herdewijn, PietChemistry & Biodiversity2007 7
cpdart0177Improved anti-osteoporosis potency and reduced endometrial membrane hyperplasia during hormone replacement therapy with estrogen-RGD peptide conjugatesXiong, Yu; Zhao, Ming; Wang, Chao; Chang, Heng Wei; Peng, ShiqiJournal of Medicinal Chemistry2007 10
cpdart0178(p-Sulfomethyl)phenylalanine as a mimic of O-sulfatyl-tyrosine in synthetic partial sequences of P-Selectin glycoprotein ligand 1 (PSGL-1)Herzner, Holger; Kunz, HorstTetrahedron2007 3
cpdart0179Synthesis and Binding Studies of Alzheimer Ligands on Solid SupportRzepecki, Petra; Geib, Nina; Peifer, Manuel; Biesemeier, Frank; Schrader, ThomasJournal of Organic Chemistry2007 9
cpdart0180Synthesis of Biologically Active Peptide Nucleic Acid-Peptide Conjugates by Sortase-Mediated LigationPritz, Stephan; Wolf, Yvonne; Kraetke, Oliver; Klose, Jana; Bienert, Michael; Beyermann, MichaelJournal of Organic Chemistry2007 20
cpdart0181A Peptide Conjugate of Vitamin E Succinate Targets Breast Cancer Cells with High ErbB2 ExpressionWang, Xiu-Fang; Birringer, Marc; Dong, Lan-Feng; Veprek, Pavel; Low, Pauline; Swettenham, Emma; Stantic, Marina; Yuan, Lin-Hong; Zobalova, Renata; Wu, Kun; Ledvina, Miroslav; Ralph, Stephen J.; Neuzil, JiriCancer Research2007 1
cpdart0182Spacer-separated sialyl Lewisx cyclo-peptide conjugates as potential E-selectin ligandsHerzner, Holger; Kunz, HorstCarbohydrate Research2007 2
cpdart0183The use of fullerene substituted phenylalanine amino acid as a passport for peptides through cell membranesYang, Jianzhong; Wang, Kuan; Driver, Jonathan; Yang, Jianhua; Barron, Andrew R.Organic & Biomolecular Chemistry2007 5
cpdart0184Bifunctional ligands that target cells displaying the αvβ3 integrinOwen, Robert M.; Carlson, Coby B.; Xu, Jinwang; Mowery, Patricia; Fasella, Elisabetta; Kiessling, Laura L.ChemBioChem2007 4
cpdart0185AZT and AZT-monophosphate prodrugs incorporating HIV-protease substrate fragment: synthesis and evaluation as specific drug delivery systemsLiotard, Jean-Francois; Mehiri, Mohamed; Di Giorgio, Audrey; Boggetto, Nicole; Reboud-Ravaux, Michele; Aubertin, Anne-Marie; Condom, Roger; Patino, NadiaAntiviral Chemistry & Chemotherapy2006 28
cpdart0186Acridin-9-yl exchange: a proposal for the action of some 9-aminoacridine drugsSebestik, Jaroslav; Safarik, Martin; Stibor, Ivan; Hlavacek, JanBiopolymers2006 2
cpdart0187REPLACE: a strategy for iterative design of cyclin-binding groove inhibitorsAndrews, Martin J. I.; Kontopidis, George; McInnes, Campbell; Plater, Andy; Innes, Lorraine; Cowan, Angela; Jewsbury, Philip; Fischer, Peter M.ChemBioChem2006 17
cpdart0188Delivery of 2-5A cargo into living cells using the Tat cell penetrating peptide: 2-5A-tatZhou, Longhu; Thakur, Chandar S.; Molinaro, Ross J.; Paranjape, Jayashree M.; Hoppes, Rieuwert; Jeang, Kuan-Teh; Silverman, Robert H.; Torrence, Paul F.Bioorganic & Medicinal Chemistry2006 4
cpdart0189Improved Therapeutic Efficacy of Doxorubicin through Conjugation with a Novel Peptide Drug Delivery Technology (Vectocell)Meyer-Losic, Florence; Quinonero, Jerome; Dubois, Vincent; Alluis, Bertrand; Dechambre, Mireille; Michel, Matthieu; Cailler, Francoise; Fernandez, Anne-Marie; Trouet, Andre; Kearsey, JonathanJournal of Medicinal Chemistry2006 7
cpdart0190Dual-acting agents that possess free radical scavenging and antithrombotic activities: Design, synthesis, and evaluation of phenolic tetrahydro-β-carboline RGD peptide conjugatesBi, Wei; Bi, Lanrong; Cai, Jianhui; Liu, Sanguang; Peng, Shiqi; Fischer, Nicholas O.; Tok, Jeffrey B.-H.; Wang, GuohuaBioorganic & Medicinal Chemistry2006 6
cpdart0191Turn and helical peptide spacers: combined distance and angular dependencies in the exciton-coupled circular dichroism of intramolecularly interacting bis-porphyrinsGuryanov, Ivan; Moretto, Alessandro; Campestrini, Sandro; Broxterman, Quirinus B.; Kaptein, Bernard; Peggion, Cristina; Formaggio, Fernando; Toniolo, ClaudioBiopolymers2006 13
cpdart0192New peptide conjugates with 9-aminoacridine: synthesis and binding to DNASebestik, Jaroslav; Stibor, Ivan; Hlavacek, JanJournal of Peptide Science2006 7
cpdart0193Single-Drug Multiligand Conjugates: Synthesis and Preliminary Cytotoxicity Evaluation of a Paclitaxel-Dipeptide "Scorpion"" Molecule"Safavy, Ahmad; Raisch, Kevin P.; Matusiak, Damien; Bhatnagar, Saloni; Helson, LawrenceBioconjugate Chemistry2006 2
cpdart0194Phosphorylation State-Responsive Lanthanide Peptide Conjugates: A Luminescence Switch Based on Reversible Complex ReorganizationTremblay, Matthew S.; Zhu, Qing; Marti, Angel A.; Dyer, Joanne; Halim, Marlin; Jockusch, Steffen; Turro, Nicholas J.; Sames, DaliborOrganic Letters2006 2
cpdart0195Synthesis of oligotuftsin-based branched oligopeptide conjugates for chemotactic drug targetingMezo, Gabor; Lang, Orsolya; Jakab, Annamaria; Bai, Katalin B.; Szabo, Ildiko; Schlosser, Gitta; Lang, Julianna; Kohidai, Laszlo; Hudecz, FerencJournal of Peptide Science2006 3
cpdart0196Peptide-doxorubicin conjugates specifically degraded by matrix metalloproteinases expressed from tumorLee, Gee Young; Song, Ji-hye; Kim, Sang Yoon; Park, Kyeongsoon; Byun, YoungroDrug Development Research2006 6
cpdart0197Synthesis and biological activity of conjugates between paclitaxel and the cell delivery vector penetratinWang, Shudong; Zhelev, Nikolai Z.; Duff, Susan; Fischer, Peter M.Bioorganic & Medicinal Chemistry2006 6
cpdart0198Design of an IV Formulation of an Unstable Prodrug Candidate for Prostate Cancer Treatment: Solution Chemistry of N-(glutaryl-hyp-ala-ser-cyclohexylglycyl-gln-ser-leu)-doxorubicinKarki, Shyam; Treemaneekarn, Varaporn; Ostovic, Drazen; Nerurkar, Maneesh; Almarsson, OernDrug Development and Industrial Pharmacy2006 1
cpdart0199Peptide-Mediated Cell Transport of Water Soluble Porphyrin ConjugatesSibrian-Vazquez, Martha; Jensen, Timothy J.; Hammer, Robert P.; Vicente, M. Graca H.Journal of Medicinal Chemistry2006 5
cpdart0200Synthesis of acridine-nuclear localization signal (NLS) conjugates and evaluation of their impact on lipoplex and polyplex-based transfectionBoulanger, Caroline; Di Giorgio, Christophe; Vierling, PierreEuropean Journal of Medicinal Chemistry2005 4
cpdart0201Synthesis and characterization of positively charged porphyrin-peptide conjugatesSibrian-Vazquez, Martha; Jensen, Timothy J.; Fronczek, Frank R.; Hammer, Robert P.; Vicente, M. Graca H.Bioconjugate Chemistry2005 10
cpdart0202Mechanism and structure-activity relationships of norspermidine-based peptidic inhibitors of trypanothione reductaseDixon, Mark J.; Maurer, Richard I.; Biggi, Cristina; Oyarzabal, Julen; Essex, Jonathan W.; Bradley, MarkBioorganic & Medicinal Chemistry2005 2
cpdart0203Synthesis and Biological Activity of Nitronyl Nitroxide Containing PeptidesZhao, Ming; Liu, Junling; Wang, Chao; Wang, Lili; Liu, Hu; Peng, ShiqiJournal of Medicinal Chemistry2005 11
cpdart0204Self-Assembling Porphyrin-Modified PeptidesDunetz, Joshua R.; Sandstrom, Claire; Young, Elizabeth R.; Baker, Paul; Van Name, Steven A.; Cathopolous, Terry; Fairman, Robert; De Paula, Julio C.; Kerfeldt, Karin S.Organic Letters2005 1
cpdart0205One pot conjugation of the polypeptides directed by phosphorus oxychlorideZhou, N.; Liu, Y.; Zhou, G. J.; Zhao, Y. F.Journal of Peptide Research2005 18
cpdart0206Synthesis, Characterization, and Cellular Uptake of DNA-Binding Rose Bengal PeptidoconjugatesCarreon, Jay R.; Roberts, Marcel A.; Wittenhagen, Lisa M.; Kelley, Shana O.Organic Letters2005 7
cpdart0207DNA scission chemistry and EPR studies of four new bis(2,6-dimethoxyhydroquinone-3-mercaptoacetic acid)-peptide conjugatesSong, Yu-FeiAustralian Journal of Chemistry2004 4
cpdart0208Synthesis of a silk-inspired peptide-oligothiophene conjugateKlok, Harm-Anton; Roesler, Annette; Goetz, Guenther; Mena-Osteritz, Elena; Baeuerle, PeterOrganic & Biomolecular Chemistry2004 1
cpdart0209Synthesis and Characterization of Peptide-Cationic Steroid Antibiotic ConjugatesDing, Bangwei; Taotofa, Uale; Orsak, Thomas; Chadwell, Matthew; Savage, Paul B.Organic Letters2004 9
cpdart0210The synthesis and immunosuppressive activities of steroid-urotoxin linkersWang, Chao; Zhao, Ming; Qiu, Xuecai; Peng, ShiqiBioorganic & Medicinal Chemistry2004 13
cpdart0211De novo design, synthesis, and function of semiartificial myoglobin conjugated with coiled-coil two-α-helix peptidesSakamoto, Seiji; Ito, Atsushi; Kudo, Kazuaki; Yoshikawa, SusumuChemistry - A European Journal2004 3
cpdart02122-Pyrrolinodoxorubicin and its peptide-vectorized form bypass multidrug resistanceCastex, Cedric; Merida, Peggy; Blanc, Emmanuelle; Clair, Philippe; Rees, Anthony R.; Temsamani, JamalAnti-Cancer Drugs2004 3
cpdart0213Arginine carrier peptide bearing Ni(II) chelator to promote cellular uptake of histidine-tagged proteinsFutaki, Shiroh; Niwa, Miki; Nakase, Ikuhiko; Tadokoro, Akiko; Zhang, Youjun; Nagaoka, Makoto; Wakako, Naoya; Sugiura, YukioBioconjugate Chemistry2004 5
cpdart0214Efficient synthesis of RGD-containing cyclic peptide-porphyrin conjugates by ring-closing metathesis on solid supportChaleix, Vincent; Sol, Vincent; Guilloton, Michel; Granet, Robert; Krausz, PierreTetrahedron Letters2004 6
cpdart0215Design, synthesis, and characterization of an ATP-peptide conjugate inhibitor of protein kinase AHines, Aliya C.; Cole, Philip A.Bioorganic & Medicinal Chemistry Letters2004 3
cpdart0216Thiazole orange-peptide conjugates: Sensitivity of DNA binding to chemical structureCarreon, Jay R.; Mahon, Kerry P. Jr.; Kelley, Shana O.Organic Letters2004 4
cpdart0217Zipper-Featured δ-Peptide Foldamers Driven by Donor-Acceptor Interaction. Design, Synthesis, and CharacterizationZhao, Xin; Jia, Mu-Xin; Jiang, Xi-Kui; Wu, Li-Zhu; Li, Zhan-Ting; Chen, Guang-JuJournal of Organic Chemistry2004 9
cpdart0218HPLC-MS/MS determination of a peptide conjugate prodrug of doxorubicin, and its active metabolites, leucine-doxorubicin and doxorubicin, in dog and rat plasmaMazuel, Claude; Grove, Jeffrey; Gerin, Genevieve; Keenan, Kevin P.Journal of Pharmaceutical and Biomedical Analysis2003 2
cpdart0219Toward Artificial Developmental RegulatorsArndt, Hans-Dieter; Hauschild, Karl E.; Sullivan, David P.; Lake, Kara; Dervan, Peter B.; Ansari, Aseem Z.Journal of the American Chemical Society2003 2
cpdart0220Receptor-Mediated Targeting of a Photosensitizer by Its Conjugation to Gonadotropin-Releasing Hormone AnaloguesRahimipour, Shai; Ben-Aroya, Nurit; Ziv, Keren; Chen, Alon; Fridkin, Mati; Koch, YitzhakJournal of Medicinal Chemistry2003 2
cpdart0221Self-Assembling of the Porphyrin-Linked Acyclic Penta- and Heptapeptides in Aqueous TrifluoroethanolArai, Toru; Inudo, Makiko; Ishimatsu, Tomomi; Akamatsu, Chieko; Tokusaki, Yasushi; Sasaki, Tomikazu; Nishino, NorikazuJournal of Organic Chemistry2003 3
cpdart0222An efficient synthesis of a doxorubicin-peptide conjugateShi, Yao-Jun; Cameron, Mark; Dolling, Ulf H.; Lieberman, David R.; Lynch, Joseph E.; Reamer, Robert A.; Robbins, Michael A.; Volante, R. P.; Reider, Paul J.Synlett2003 1
cpdart0223New dsDNA-binding hybrid molecules combining an unnatural peptide and an intercalating moietyChaltin, Patrick; Borgions, Filip; Rozenski, Jef; Van Aerschot, Arthur; Herdewijn, PietHelvetica Chimica Acta2003 23
cpdart0224An adjustable release rate linking strategy for cytotoxin-Peptide conjugates Fuselier, Joseph A.; Sun, Lichun; Woltering, S. Nathaniel; Murphy, William A.; Vasilevich, Natalya; Coy, David H.Bioorganic & Medicinal Chemistry Letters2003 6
cpdart0225Amino acid and peptide conjugates of protoporphyrin: preparation and analysis by high-performance liquid chromatography, high-performance liquid chromatography/electrospray ionization mass spectrometry and matrix-assisted laser desorption/ionization time-of-flight mass spectrometryRazzaque, M. A.; Lord, G. A.; Lim, C. K.Rapid Communications in Mass Spectrometry2002 7
cpdart0226DNA Cross-Linking with Metallointercalator-Peptide ConjugatesCopeland, Kimberly D.; Lueras, Alexis M. K.; Stemp, Eric D. A.; Barton, Jacqueline K.Biochemistry2002 12
cpdart0227Investigations into the chromatographic behavior of a doxorubicin-peptide conjugateHicks, Michael B.; Antonucci, Vincent L.; Riddle, Lance; Novak, Tom J.; Skrdla, PeterJournal of Chromatography A2002 1
cpdart0228Design and Synthesis of a Pro-Drug of Vinblastine Targeted at Treatment of Prostate Cancer with Enhanced Efficacy and Reduced Systemic ToxicityBrady, Stephen F.; Pawluczyk, Joseph M.; Lumma, Patricia K.; Feng, Dong-Mei; Wai, Jenny M.; Jones, Raymond; DeFeo-Jones, Deborah; Wong, Bradley K.; Miller-Stein, Cynthia; Lin, Jiunn H.; Oliff, Allen; Freidinger, Roger M.; Garsky, Victor M.Journal of Medicinal Chemistry2002 5
cpdart0229Advanced Synthesis & CatalysisMann, Enrique; Chana, Antonio; Sanchez-Sancho, Francisco; Puerta, Carmen; Garcia-Merino, Antonio; Herradon, BernardoAdvanced Synthesis & Catalysis2002 9
cpdart0230Solid-Phase Synthesis of Symmetrical 3,6-Bispeptide-Acridone ConjugatesLadame, Sylvain; Harrison, R. John; Neidle, Stephen; Balasubramanian, ShankarOrganic Letters2002 4
cpdart0231Employment of on-line FT-IR spectroscopy to monitor the deprotection of a 9-fluorenylmethyl protected carboxylic acid peptide conjugate of doxorubicinCameron, Mark; Zhou, George X.; Hicks, Micheal B.; Antonucci, Vincent; Ge, Zhihong; Lieberman, David R.; Lynch, Joesph E.; Shi, Yao-JunJournal of Pharmaceutical and Biomedical Analysis2002 4
cpdart0232Characterization of a novel prostate-specific antigen-activated peptide-doxorubicin conjugate in patients with prostate cancerDiPaola, Robert S.; Rinehart, John; Nemunaitis, John; Ebbinghaus, Scott; Rubin, Eric; Capanna, Terry; Ciardella, Marie; Doyle-Lindrud, Susan; Goodwin, Susan; Fontaine, Michelle; Adams, Ned; Williams, Adrienne; Schwartz, Michael; Winchell, Greg; Wickersham, Karen; Deutsch, Paul; Yao, Siu-LongJournal of Clinical Oncology2002 1
cpdart0233Targeted Type 1 phototherapeutic agents using azido-peptide bioconjugatesRajagopalan, Raghavan; Achilefu, Samuel I.; Jimenez, Hermo N.; Webb, Elizabeth G.; Schmidt, Michelle A.; Bugaj, Joseph E.; Dorshow, Richard B.International Society for Optical Engineering2001 5
cpdart0234Preparative Biochemistry & BiotechnologySong, Y. F.; Yang, P.Preparative Biochemistry & Biotechnology2001 8
cpdart0235The Synthesis of a Prodrug of Doxorubicin Designed to Provide Reduced Systemic Toxicity and Greater Target EfficacyGarsky, Victor M.; Lumma, Patricia K.; Feng, Dong-Mei; Wai, Jenny; Ramjit, Harri G.; Sardana, Mohinder K.; Oliff, Allen; Jones, Raymond E.; DeFeo-Jones, Deborah; Freidinger, Roger M.Journal of Medicinal Chemistry2001 13
cpdart0236Improvement of Porphyrin Cellular Delivery and Activity by Conjugation to a Carrier PeptideChaloin, Laurent; Bigey, Pascal; Loup, Christophe; Marin, Mariana; Galeotti, Nathalie; Piechaczyk, Marc; Heitz, Frederic; Meunier, BernardBioconjugate Chemistry2001 2
cpdart0237Anthraquinone-peptides as inhibitors of AP-1 transcription factorIjaz, T.; Tran, P.; Ruparelia, K. C.; Teesdale-Spittle, P. H.; Orr, S.; Patterson, L. H.Bioorganic & Medicinal Chemistry Letters2001 8
cpdart0238Determinants for the drug release from T-0128, camptothecin analog-carboxymethyl dextran conjugateHarada, M.; Sakakibara, H.; Yano, T.; Suzuki, T.; Okuno, S.Journal of Controlled Release2000 9
cpdart0239Preparation and biological activity of amino acid and peptide conjugates of antitumor hydroxymethylacylfulveneMcMorris, Trevor C.; Yu, Jian; Ngo, Huan-Tony; Wang, Haixia; Kelner, Michael J.Journal of Medicinal Chemistry2000 4
cpdart0240Solid-phase synthesis of acridine-peptide conjugates and their analysis by tandem mass spectrometryCarlson, Coby B.; Beal, Peter A.Organic Letters2000 3
cpdart0241Highly parallel nano-synthesis of cleavable peptide-dye conjugates on cellulose membranesLicha, Kai; Bhargava, Sarah; Rheinlander, Christiane; Becker, Andreas; Schneider-Mergener, Jens; Volkmer-Engert, RudolfTetrahedron Letters2000 2
cpdart0242Synthesis of porphyrin α,ω-bis(methylamino)peptide constructsMatthews, Susan E.; Pouton, Colin W.; Threadgill, Michael D.New Journal of Chemistry1999 9
cpdart0243Cancer chemotherapy based on targeting of cytotoxic peptide conjugates to their receptors on tumorsSchally, Andrew V.; Nagy, AttilaEuropean Journal of Endocrinology1999 1
cpdart0244Synthesis of the palmitoylated and prenylated C-terminal lipopeptides of the human R- and N-Ras proteinsSchmittberger, T.; Waldmann, H.Bioorganic & Medicinal Chemistry1999 20
cpdart0245A calixarene with four peptide loops: an antibody mimic for recognition of protein surfacesHamuro, Yoshitomo; Calama, Mercedes Crego; Park, Hyung Soon; Hamilton, Andrew D.Angewandte Chemie, International Edition in English1997 4
cpdart0246Benzenesulfonamide-peptide conjugates as probes for secondary binding sites near the active site of carbonic anhydraseSigal, George B.; Whitesides, George M.Bioorganic & Medicinal Chemistry Letters1996 43
cpdart0247Synthesis of carboxymethylpullulan-peptide-doxorubicin conjugates and their propertiesNogusa, Hideo; Yano, Toshiro; Okuno, Satoshi; Hamana, Hiroshi; Inoue, KazuhiroChemical & Pharmaceutical Bulletin1995 1
cpdart0248Synthesis and immunological evaluation of the conjugates composed of a muramyl peptide GMDP and tuftsinTitov, Vladimir M.; Meshcheryakova, Elena A.; Balashova, Tamara A.; Andronova, Tatyana M.; Ivanov, Vadim T.International Journal of Peptide & Protein Research1995 4
cpdart0249A Bioactive Fullerene PeptideToniolo, Claudio; Bianco, Alberto; Maggini, Michele; Scorrano, Gianfranco; Prato, Maurizio; Marastoni, Mauro; Tomatis, Roberto; Spisani, Susanna; Palu, Giorgio; Blair, Edward D.Journal of Medicinal Chemistry1994 1
cpdart0250Preparation of Vitamin B6-Conjugated Peptides at the Amino Terminus and of Vitamin B6-Peptide-Oligonucleotide ConjugatesZhu, Tianmin; Stein, StanleyBioconjugate Chemistry1994 1
cpdart0251Studies of N-terminal templates for α-helix formation. Synthesis and conformational analysis of peptide conjugates of (2S,5S,8S,11S)-1-acetyl-1,4-diaza-3-keto-5-carboxy-10-thiatricyclo[2.8.1.04,8]tridecane (Ac-Hel1-OH)Kemp, D. S.; Curran, Timothy P.; Boyd, James G.; Allen, Thomas J.Journal of Organic Chemistry1991 10